PDB entry 3vbw
View 3vbw on RCSB PDB site
Description: Exploitation of hydrogen bonding constraints and flat hydrophobic energy landscapes in Pim-1 kinase needle screening and inhibitor design
Class: transferase/transferase inhibitor
Keywords: Pim1, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-01-02, released
2012-03-21
The last revision prior to the SCOPe 2.06 freeze date was dated
2012-05-16, with a file datestamp of
2012-05-11.
Experiment type: XRAY
Resolution: 2.48 Å
R-factor: 0.232
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase pim-1
Species: Homo sapiens [TaxId:9606]
Gene: PIM1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3vbwa_ - Heterogens: 0FN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3vbwA (A:)
mkekeplesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvp
mevvllkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsf
fwqvleavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvy
sppewiryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhli
rwclalrpsdrptfeeiqnhpwmqdvllpqetaeihlhslspgpskaaalehhhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3vbwA (A:)
esqyqvgpllggsvysgirvsdnlpvaikhvekdrisdwgeltrvpmevvllkkvssgfs
gvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvleavrhchnc
gvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppewiryhryhgr
saavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwclalrpsdrptf
eeiqnhpwmqdvllpqetaeihlh