PDB entry 3uli
View 3uli on RCSB PDB site
Description: Human Cyclin Dependent Kinase 2 (CDK2) bound to azabenzimidazole derivative
Class: transferase/transferase inhibitor
Keywords: azabenzimidazole derivative, Phosphotransfer, Complex with Cyclin A or Cyclin E, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-11-10, released
2013-08-14
The last revision prior to the SCOPe 2.08 freeze date was dated
2013-09-04, with a file datestamp of
2013-08-30.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.238
AEROSPACI score: 0.39
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cyclin-dependent kinase 2
Species: Homo sapiens [TaxId:9606]
Gene: CDK2, CDKN2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3ulia_ - Heterogens: 1N3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3uliA (A:)
menfqkvekigegtygvvykarnkltgevvalkkirldtetegvpstaireisllkelnh
pnivklldvihtenklylvfeflhqdlkkfmdasaltgiplpliksylfqllqglafchs
hrvlhrdlkpqnllintegaikladfglarafgvpvrtythevvtlwyrapeillgckyy
stavdiwslgcifaemvtrralfpgdseidqlfrifrtlgtpdevvwpgvtsmpdykpsf
pkwarqdfskvvppldedgrsllsqmlhydpnkrisakaalahpffqdvtkpvphlrl
Sequence, based on observed residues (ATOM records): (download)
>3uliA (A:)
menfqkvekigegtygvvykarnkltgevvalkkirldvpstaireisllkelnhpnivk
lldvihtenklylvfeflhqdlkkfmdasaltgiplpliksylfqllqglafchshrvlh
rdlkpqnllintegaikladfglarafgvevvtlwyrapeillgckyystavdiwslgci
faemvtrralfpgdseidqlfrifrtlgtpdevvwpgvtsmpdykpsfpkwarqdfskvv
ppldedgrsllsqmlhydpnkrisakaalahpffqdvtkpvphlrl