PDB entry 3uhl
View 3uhl on RCSB PDB site
Description: Crystal Structure of Multidrug Resistant HIV-1 Protease Clinical Isolate PR20 in Complex with p2-NC substrate analog
Class: Hydrolase/Hydrolase inhibitor
Keywords: Hydrolase-Hydrolase inhibitor complex
Deposited on
2011-11-03, released
2012-03-28
The last revision prior to the SCOPe 2.04 freeze date was dated
2012-10-17, with a file datestamp of
2012-10-12.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.231
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot P03367 (0-98)
- engineered mutation (6)
- engineered mutation (9)
- engineered mutation (12)
- engineered mutation (14)
- engineered mutation (29)
- engineered mutation (31-32)
- engineered mutation (34-36)
- engineered mutation (46)
- engineered mutation (53)
- engineered mutation (57)
- engineered mutation (61-62)
- engineered mutation (66)
- engineered mutation (70)
- engineered mutation (83)
- engineered mutation (87-89)
- engineered mutation (94)
Domains in SCOPe 2.04: d3uhla_ - Chain 'B':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot P03367 (0-98)
- engineered mutation (6)
- engineered mutation (9)
- engineered mutation (12)
- engineered mutation (14)
- engineered mutation (29)
- engineered mutation (31-32)
- engineered mutation (34-36)
- engineered mutation (46)
- engineered mutation (53)
- engineered mutation (57)
- engineered mutation (61-62)
- engineered mutation (66)
- engineered mutation (70)
- engineered mutation (83)
- engineered mutation (87-89)
- engineered mutation (94)
Domains in SCOPe 2.04: d3uhlb_ - Chain 'C':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot P03367 (0-98)
- engineered mutation (6)
- engineered mutation (9)
- engineered mutation (12)
- engineered mutation (14)
- engineered mutation (29)
- engineered mutation (31-32)
- engineered mutation (34-36)
- engineered mutation (46)
- engineered mutation (53)
- engineered mutation (57)
- engineered mutation (61-62)
- engineered mutation (66)
- engineered mutation (70)
- engineered mutation (83)
- engineered mutation (87-89)
- engineered mutation (94)
Domains in SCOPe 2.04: d3uhlc_ - Chain 'D':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot P03367 (0-98)
- engineered mutation (6)
- engineered mutation (9)
- engineered mutation (12)
- engineered mutation (14)
- engineered mutation (29)
- engineered mutation (31-32)
- engineered mutation (34-36)
- engineered mutation (46)
- engineered mutation (53)
- engineered mutation (57)
- engineered mutation (61-62)
- engineered mutation (66)
- engineered mutation (70)
- engineered mutation (83)
- engineered mutation (87-89)
- engineered mutation (94)
Domains in SCOPe 2.04: d3uhld_ - Heterogens: SO4, 2NC, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>3uhlA (A:)
pqitlwkrpfvtvkvggqlkealldtgadntifedinlpgrwkpkmvggiggflkvreyd
qvpieiaghkvigtvlvgptpvnvigrdtmtqigatlnf
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>3uhlB (B:)
pqitlwkrpfvtvkvggqlkealldtgadntifedinlpgrwkpkmvggiggflkvreyd
qvpieiaghkvigtvlvgptpvnvigrdtmtqigatlnf
- Chain 'C':
Sequence; same for both SEQRES and ATOM records: (download)
>3uhlC (C:)
pqitlwkrpfvtvkvggqlkealldtgadntifedinlpgrwkpkmvggiggflkvreyd
qvpieiaghkvigtvlvgptpvnvigrdtmtqigatlnf
- Chain 'D':
Sequence; same for both SEQRES and ATOM records: (download)
>3uhlD (D:)
pqitlwkrpfvtvkvggqlkealldtgadntifedinlpgrwkpkmvggiggflkvreyd
qvpieiaghkvigtvlvgptpvnvigrdtmtqigatlnf