PDB entry 3u51
View 3u51 on RCSB PDB site
Description: Src in complex with DNA-templated macrocyclic inhibitor MC1
Class: transferase/transferase inhibitor
Keywords: protein kinase, Src-like inactive conformation, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-10-10, released
2012-02-22
The last revision prior to the SCOPe 2.04 freeze date was dated
2012-04-04, with a file datestamp of
2012-03-30.
Experiment type: XRAY
Resolution: 2.24 Å
R-factor: 0.2
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Proto-oncogene tyrosine-protein kinase Src
Species: Gallus gallus [TaxId:9031]
Gene: SRC
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d3u51a_ - Chain 'B':
Compound: Proto-oncogene tyrosine-protein kinase Src
Species: Gallus gallus [TaxId:9031]
Gene: SRC
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d3u51b_ - Heterogens: 08X, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3u51A (A:)
aweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaflqeaqvmkklr
heklvqlyavvseepiyivteymskgslldflkgemgkylrlpqlvdmaaqiasgmayve
rmnyvhrdlraanilvgenlvckvadfglarliedneytarqgakfpikwtapeaalygr
ftiksdvwsfgilltelttkgrvpypgmvnrevldqvergyrmpcppecpeslhdlmcqc
wrkdpeerptfeylqafledyftstepqyqpgenl
Sequence, based on observed residues (ATOM records): (download)
>3u51A (A:)
eipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaflqeaqvmkklrhe
klvqlyavvseepiyivteymskgslldflkgemgkylrlpqlvdmaaqiasgmayverm
nyvhrdlraanilvgenlvckvadfgfpikwtapeaalygrftiksdvwsfgillteltt
kgrvpypgmvnrevldqvergyrmpcppecpeslhdlmcqcwrkdpeerptfeylqafle
dyftstepqyqpgenl
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3u51B (B:)
aweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaflqeaqvmkklr
heklvqlyavvseepiyivteymskgslldflkgemgkylrlpqlvdmaaqiasgmayve
rmnyvhrdlraanilvgenlvckvadfglarliedneytarqgakfpikwtapeaalygr
ftiksdvwsfgilltelttkgrvpypgmvnrevldqvergyrmpcppecpeslhdlmcqc
wrkdpeerptfeylqafledyftstepqyqpgenl
Sequence, based on observed residues (ATOM records): (download)
>3u51B (B:)
eipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaflqeaqvmkklrhe
klvqlyavvseepiyivteymskgslldflkgemgkylrlpqlvdmaaqiasgmayverm
nyvhrdlraanilvgenlvckvadfgpikwtapeaalygrftiksdvwsfgilltelttk
grvpypgmvnrevldqvergyrmpcppecpeslhdlmcqcwrkdpeerptfeylqafled
yftstepqyqpgenl