PDB entry 3u2o
View 3u2o on RCSB PDB site
Description: Dihydroorotate Dehydrogenase (DHODH) crystal structure in complex with small molecule inhibitor
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: DHODH, DEHYDROGENASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on
2011-10-04, released
2011-11-16
The last revision prior to the SCOPe 2.07 freeze date was dated
2012-09-05, with a file datestamp of
2012-08-31.
Experiment type: XRAY
Resolution: 2.18 Å
R-factor: 0.161
AEROSPACI score: 0.44
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dihydroorotate dehydrogenase (quinone), mitochondrial
Species: Homo sapiens [TaxId:9606]
Gene: DHODH
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d3u2oa_ - Heterogens: FMN, ORO, 03U, ACT, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3u2oA (A:)
mawrhlkkraqdaviilggggllfasylmatgderfyaehlmptlqglldpesahrlavr
ftslgllprarfqdsdmlevrvlghkfrnpvgiaagfdkhgeavdglykmgfgfveigsv
tpkpqegnprprvfrlpedqavinrygfnshglsvvehrlrarqqkqakltedglplgvn
lgknktsvdaaedyaegvrvlgpladylvvnvsspntaglrslqgkaelrrlltkvlqer
dglrrvhrpavlvkiapdltsqdkediasvvkelgidglivtnttvsrpaglqgalrset
gglsgkplrdlstqtiremyaltqgrvpiigvggvssgqdalekiragaslvqlytaltf
wgppvvgkvkreleallkeqgfggvtdaigadhrr
Sequence, based on observed residues (ATOM records): (download)
>3u2oA (A:)
matgderfyaehlmptlqglldpesahrlavrftslgllprarfqdsdmlevrvlghkfr
npvgiaagfdkhgeavdglykmgfgfveigsvtpkpqegnprprvfrlpedqavinrygf
nshglsvvehrlrarqqkqakltedglplgvnlgknktsvdaaedyaegvrvlgpladyl
vvnvsspntaglrslqgkaelrrlltkvlqerdglrrvhrpavlvkiapdltsqdkedia
svvkelgidglivtnttvsrpaglqgalrsetgglsgkplrdlstqtiremyaltqgrvp
iigvggvssgqdalekiragaslvqlytaltfwgppvvgkvkreleallkeqgfggvtda
igadhr