PDB entry 3she
View 3she on RCSB PDB site
Description: Novel ATP-competitive MK2 inhibitors with potent biochemical and cell-based activity throughout the series
Class: transferase/transferase inhibitor
Keywords: Kinase domain with bound inhibitor, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-06-16, released
2011-12-14
The last revision prior to the SCOPe 2.08 freeze date was dated
2012-01-11, with a file datestamp of
2012-01-06.
Experiment type: XRAY
Resolution: 2.25 Å
R-factor: 0.248
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: MAP kinase-activated protein kinase 3
Species: Homo sapiens [TaxId:9606]
Gene: MAPKAPK3
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3shea_ - Heterogens: I85, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3sheA (A:)
epkkyavtddyqlskqvlglgvngkvlecfhrrtgqkcalkllydspkarqevdhhwqas
ggphivcildvyenmhhgkrclliimecmeggelfsriqergdqaftereaaeimrdigt
aiqflhshniahrdvkpenllytskekdavlkltdfgfakettqnalqtpcytpyyvape
vlgpekydkscdmwslgvimyillcgfppfysntgqaispgmkrrirlgqygfpnpewse
vsedakqlirlllktdpterltitqfmnhpwinqsmvvpqtplhtarvlqedkdhwdevk
eemtsalatmrvdydqv
Sequence, based on observed residues (ATOM records): (download)
>3sheA (A:)
epkkyavtddyqlskqvlglgvngkvlecfhrrtgqkcalkllydspkarqevdhhwqas
ggphivcildvyenmhhgkrclliimecmeggelfsriqeaftereaaeimrdigtaiqf
lhshniahrdvkpenllytskekdavlkltdfgfaketekydkscdmwslgvimyillcg
fppfygfpnpewsevsedakqlirlllktdpterltitqfmnhpwinqsmvvpqtplhta
rvlqedkdhwdevkeemtsalatmrvdydq