PDB entry 3s56
View 3s56 on RCSB PDB site
Description: HIV-1 protease triple mutants V32I, I47V, V82I with antiviral drug saquinavir
Class: hydrolase/hydrolase inhibitor
Keywords: SAQUINAVIR,HIV/AIDS, drug resistance, aspartic protease, molecular recognition, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2011-05-20, released
2012-03-21
The last revision prior to the SCOPe 2.08 freeze date was dated
2012-03-21, with a file datestamp of
2012-03-16.
Experiment type: XRAY
Resolution: 1.88 Å
R-factor: 0.188
AEROSPACI score: 0.47
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot Q7SSI0 (0-98)
- engineered mutation (6)
- engineered mutation (31-32)
- engineered mutation (46)
- engineered mutation (62)
- engineered mutation (66)
- engineered mutation (81)
- engineered mutation (94)
Domains in SCOPe 2.08: d3s56a_ - Chain 'B':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot Q7SSI0 (0-98)
- engineered mutation (6)
- engineered mutation (31-32)
- engineered mutation (46)
- engineered mutation (62)
- engineered mutation (66)
- engineered mutation (81)
- engineered mutation (94)
Domains in SCOPe 2.08: d3s56b_ - Heterogens: ROC, ACT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>3s56A (A:)
pqitlwkrplvtikiggqlkealldtgaddtiieemslpgrwkpkmvggiggfikvrqyd
qiiieiaghkaigtvlvgptpiniigrnlltqigatlnf
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>3s56B (B:)
pqitlwkrplvtikiggqlkealldtgaddtiieemslpgrwkpkmvggiggfikvrqyd
qiiieiaghkaigtvlvgptpiniigrnlltqigatlnf