PDB entry 3s4q
View 3s4q on RCSB PDB site
Description: P38 alpha kinase complexed with a pyrazolo-triazine based inhibitor
Class: transferase/transferase inhibitor
Keywords: P38 MAP KINASE, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-05-20, released
2012-02-01
The last revision prior to the SCOPe 2.08 freeze date was dated
2012-02-01, with a file datestamp of
2012-01-27.
Experiment type: XRAY
Resolution: 2.27 Å
R-factor: 0.26
AEROSPACI score: 0.26
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: CSBP, CSBP1, CSBP2, CSPB1, MAPK14, MXI2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3s4qa_ - Heterogens: NK0, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3s4qA (A:)
mahhhhhsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkk
lsrpfqsiihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadln
nivkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarh
tddemtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlkl
ilrlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsd
kritaaqalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppld
qeemes
Sequence, based on observed residues (ATOM records): (download)
>3s4qA (A:)
erptfyrqelnktiwevperyqnlspvgsvcaafdtktglrvavkklsrpfqsiihakrt
yrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivqkltddhvqfl
iyqilrglkyihsadiihrdlkpsnlavnedcelkildfglaatrwyrapeimynqtvdi
wsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqsltqmp
kmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadpydqs
fesrdllidewksltydevisfvppp