PDB entry 3s2v
View 3s2v on RCSB PDB site
Description: Crystal Structure of the Ligand Binding Domain of GluK1 in Complex with an Antagonist (S)-1-(2'-Amino-2'-carboxyethyl)-3-[(2-carboxythien-3-yl)methyl]thieno[3,4-d]pyrimidin-2,4-dione at 2.5 A Resolution
Class: membrane protein
Keywords: antagonist, Ionotropic Glutamate Receptor, MEMBRANE PROTEIN
Deposited on
2011-05-17, released
2011-06-22
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-11-08, with a file datestamp of
2017-11-03.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: N/A
AEROSPACI score: 0.2
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Glutamate receptor, ionotropic kainate 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Grik1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3s2va_ - Chain 'B':
Compound: Glutamate receptor, ionotropic kainate 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Grik1
Database cross-references and differences (RAF-indexed):
- Uniprot P22756 (1-115)
- expression tag (0)
- linker (116-117)
- Uniprot P22756 (118-256)
Domains in SCOPe 2.08: d3s2vb1, d3s2vb2 - Heterogens: 3HU, SO4, GOL, CL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3s2vA (A:)
ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
gklhmmkekwwrgngcp
Sequence, based on observed residues (ATOM records): (download)
>3s2vA (A:)
rtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkyga
qndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsa
ddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvltt
dyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegkl
hmmkekwwrgngcp
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>3s2vB (B:)
ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
gklhmmkekwwrgngcp