PDB entry 3s2v

View 3s2v on RCSB PDB site
Description: Crystal Structure of the Ligand Binding Domain of GluK1 in Complex with an Antagonist (S)-1-(2'-Amino-2'-carboxyethyl)-3-[(2-carboxythien-3-yl)methyl]thieno[3,4-d]pyrimidin-2,4-dione at 2.5 A Resolution
Class: membrane protein
Keywords: antagonist, Ionotropic Glutamate Receptor, MEMBRANE PROTEIN
Deposited on 2011-05-17, released 2011-06-22
The last revision prior to the SCOPe 2.08 freeze date was dated 2017-11-08, with a file datestamp of 2017-11-03.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: N/A
AEROSPACI score: 0.2 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Glutamate receptor, ionotropic kainate 1
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Grik1
    Database cross-references and differences (RAF-indexed):
    • Uniprot P22756 (Start-115)
      • linker (116-117)
    • Uniprot P22756 (118-256)
    Domains in SCOPe 2.08: d3s2va_
  • Chain 'B':
    Compound: Glutamate receptor, ionotropic kainate 1
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Grik1
    Database cross-references and differences (RAF-indexed):
    • Uniprot P22756 (1-115)
      • expression tag (0)
      • linker (116-117)
    • Uniprot P22756 (118-256)
    Domains in SCOPe 2.08: d3s2vb1, d3s2vb2
  • Heterogens: 3HU, SO4, GOL, CL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3s2vA (A:)
    ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
    ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
    dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
    lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
    gklhmmkekwwrgngcp
    

    Sequence, based on observed residues (ATOM records): (download)
    >3s2vA (A:)
    rtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkyga
    qndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsa
    ddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvltt
    dyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegkl
    hmmkekwwrgngcp
    

  • Chain 'B':
    Sequence; same for both SEQRES and ATOM records: (download)
    >3s2vB (B:)
    ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
    ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
    dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
    lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
    gklhmmkekwwrgngcp