PDB entry 3r2y
View 3r2y on RCSB PDB site
Description: MK2 kinase bound to Compound 1
Class: transferase/transferase inhibitor
Keywords: Kinase domain, Phosphotransferase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-03-15, released
2011-05-25
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-07-13, with a file datestamp of
2011-07-08.
Experiment type: XRAY
Resolution: 3 Å
R-factor: 0.294
AEROSPACI score: 0.13
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: MAP kinase-activated protein kinase 2
Species: Homo sapiens [TaxId:9606]
Gene: MAPKAPK2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3r2ya_ - Heterogens: MLI, P4O, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3r2yA (A:)
fhvksglqikknaiiddykvtsqvlglgingkvlqifnkrtqekfalkmlqdcpkarrev
elhwrasqcphivrivdvyenlyagrkcllivmecldggelfsriqdrgdqafterease
imksigeaiqylhsiniahrdvkpenllytskrpnailkltdfgfakettshnslttpcy
tpyyvapevlgpekydkscdmwslgvimyillcgyppfysnhglaispgmktrirmgqye
fpnpewsevseevkmlirnllkteptqrmtitefmnhpwimqstkvpqtplhtsrvlked
kerwedvkeemtsalatmr
Sequence, based on observed residues (ATOM records): (download)
>3r2yA (A:)
fhvksglqikknaiiddykvtsqvlglgingkvlqifnkrtqekfalkmlqdcpkarrev
elhwrasqcphivrivdvyenlyagrkcllivmecldggelfsriqdtereaseimksig
eaiqylhsiniahrdvkpenllytskrpnailkltdfgfakettdkscdmwslgvimyil
lcgyppfymktrirmgqyefpnpewsevseevkmlirnllkteptqrmtitefmnhpwim
qstkvpqtplhtsrvlked