PDB entry 3qyw
View 3qyw on RCSB PDB site
Description: Crystal structure of ERK2 in complex with an inhibitor
Class: transferase/transferase inhibitor
Keywords: TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING CELL CYCLE, PHOSPHORYLATION, Protein Kinase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-03-04, released
2011-08-24
The last revision prior to the SCOPe 2.05 freeze date was dated
2012-03-21, with a file datestamp of
2012-03-16.
Experiment type: XRAY
Resolution: 1.5 Å
R-factor: 0.15
AEROSPACI score: 0.67
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Mapk1, Erk2, Mapk, Prkm1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3qywa_ - Heterogens: 6PB, DMS, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3qywA (A:)
hhhhhhmaaaaaagpemvrgqvfdvgprytnlsyigegaygmvcsaydnlnkvrvaikki
spfehqtycqrtlreikillrfrheniigindiiraptieqmkdvyivqdlmetdlykll
ktqhlsndhicyflyqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadp
dhdhtgflteyvatrwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkhyldq
lnhilgilgspsqedlnciinlkarnyllslphknkvpwnrlfpnadskaldlldkmltf
nphkrieveqalahpyleqyydpsdepiaeapfkfdmelddlpkeklkelifeetarfqp
gyrs
Sequence, based on observed residues (ATOM records): (download)
>3qywA (A:)
pemvrgqvfdvgprytnlsyigegaygmvcsaydnlnkvrvaikkispfehqtycqrtlr
eikillrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyfl
yqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadpdhdhtgflteyvat
rwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsqe
dlnciinlkarnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqalah
pyleqyydpsdepiaeapfkfdlpkeklkelifeetarfqp