PDB entry 3qlf
View 3qlf on RCSB PDB site
Description: Crystal structure of the L317I mutant of the C-src tyrosine kinase domain complexed with pyrazolopyrimidine 5
Class: transferase
Keywords: c-src l317i mutant, tyrosine kinase, transferase, pyrazolopyrimidine 5
Deposited on
2011-02-02, released
2012-02-08
The last revision prior to the SCOPe 2.03 freeze date was dated
2012-02-08, with a file datestamp of
2012-02-03.
Experiment type: XRAY
Resolution: 2.75 Å
R-factor: 0.194
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Proto-oncogene tyrosine-protein kinase Src
Species: Gallus gallus [TaxId:9031]
Gene: SRC
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3qlfa_ - Chain 'B':
Compound: Proto-oncogene tyrosine-protein kinase Src
Species: Gallus gallus [TaxId:9031]
Gene: SRC
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3qlfb_ - Heterogens: PD5, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3qlfA (A:)
ghmqtqglakdaweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaf
lqeaqvmkkirheklvqlyavvseepiyivteymskgslldflkgemgkylrlpqlvdma
aqiasgmayvermnyvhrdlraanilvgenlvckvadfglarliedneytarqgakfpik
wtapeaalygrftiksdvwsfgilltelttkgrvpypgmvnrevldqvergyrmpcppec
peslhdlmcqcwrkdpeerptfeylqafledyftstepqyqpgenl
Sequence, based on observed residues (ATOM records): (download)
>3qlfA (A:)
daweipreslrlevklgqgcfgevwmgtwngttrvaiktlklqeaqvmkkirheklvqly
avvseepiyivteymskgslldflkgemgkylrlpqlvdmaaqiasgmayvermnyvhrd
lraanilvgenlvckvadffpikwtapeaalygrftiksdvwsfgilltelttkgrvpyp
gmvnrevldqvergyrmpcppecpeslhdlmcqcwrkdpeerptfeylqafledyftste
pqyqpgenl
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3qlfB (B:)
ghmqtqglakdaweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaf
lqeaqvmkkirheklvqlyavvseepiyivteymskgslldflkgemgkylrlpqlvdma
aqiasgmayvermnyvhrdlraanilvgenlvckvadfglarliedneytarqgakfpik
wtapeaalygrftiksdvwsfgilltelttkgrvpypgmvnrevldqvergyrmpcppec
peslhdlmcqcwrkdpeerptfeylqafledyftstepqyqpgenl
Sequence, based on observed residues (ATOM records): (download)
>3qlfB (B:)
daweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpmspeaflqeaqvmkkirh
eklvqlyavvseepiyivteymskgslldflkgemgkylrlpqlvdmaaqiasgmayver
mnyvhrdlraanilvgenlvckvadfarfpikwtapeaalygrftiksdvwsfgilltel
ttkgrvpypgmvnrevldqvergyrmpcppecpeslhdlmcqcwrkdpeerptfeylqaf
ledyftstepqyqpgenl