PDB entry 3qcq
View 3qcq on RCSB PDB site
Description: Phosphoinositide-Dependent Kinase-1 (PDK1) kinase domain with 6-(3-Amino-1H-indazol-6-yl)-N4-ethyl-2,4-pyrimidinediamine
Class: transferase/transferase inhibitor
Keywords: protein-ligand complex, Kinase, Signal transduction, ATP binding Phosphoinositide binding for full length, Phoshorylation on S241, celluar and membrane associated, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-01-17, released
2011-03-09
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-03-30, with a file datestamp of
2011-03-25.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.181
AEROSPACI score: 0.36
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 3-phosphoinositide-dependent protein kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: PDK1, PDPK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3qcqa_ - Heterogens: GOL, SO4, 3Q0, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3qcqA (A:)
gpamdgtaaeprpgagslqhaqpppqprkkrpedfkfgkilgegsfstvvlarelatsre
yaikilekrhiikenkvpyvtrerdvmsrldhpffvklyftfqddeklyfglsyakngel
lkyirkigsfdetctrfytaeivsaleylhgkgiihrdlkpenillnedmhiqitdfgta
kvlspeskqaransfvgtaqyvspellteksackssdlwalgciiyqlvaglppfragne
ylifqkiikleydfpekffpkardlvekllvldatkrlgceemegygplkahpffesvtw
enlhqqtppklt
Sequence, based on observed residues (ATOM records): (download)
>3qcqA (A:)
qprkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerd
vmsrldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsa
leylhgkgiihrdlkpenillnedmhiqitdfgtakvlssfvgtaqyvspellteksack
ssdlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlvekllvlda
tkrlgceemegygplkahpffesvtwenlhqqtppkl