PDB entry 3qcj
View 3qcj on RCSB PDB site
Description: Human receptor protein tyrosine phosphatase gamma, domain 1, in complex with 5-[({3-[(3,4-dichlorobenzyl)sulfanyl]thiophen-2-yl}carbonyl)sulfamoyl]-2-methoxybenzoic acid
Class: hydrolase/hydrolase inhibitor
Keywords: TYROSINE RECEPTOR PHOSPHATASE, TWISTED MIXED BETA-SHEETS FLANKED BY {ALPHA}-HELICES, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2011-01-16, released
2011-12-28
The last revision prior to the SCOPe 2.05 freeze date was dated
2011-12-28, with a file datestamp of
2011-12-23.
Experiment type: XRAY
Resolution: 2.26 Å
R-factor: 0.215
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Receptor-type tyrosine-protein phosphatase gamma
Species: Homo sapiens [TaxId:9606]
Gene: PTPG, PTPRG
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3qcja_ - Heterogens: NX4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3qcjA (A:)
gshmgsmeaipvkqfvkhigelysnnqhgfsedfeevqrctadmnitaehsnhpenkhkn
ryinilaydhsrvklrplpgkdskhsdyinanyvdgynkakayiatqgplkstfedfwrm
iweqntgiivmitnlvekgrrkcdqywptenseeygniivtlkstkihacytvrrfsirn
tkvkkgqkgnpkgrqnervviqyhytqwpdmgvpeyalpvltfvrrssaarmpetgpvlv
hcsagvgrtgtyividsmlqqikdkstvnvlgflkhirtqrnylvqteeqyifihdalle
ailgketevs
Sequence, based on observed residues (ATOM records): (download)
>3qcjA (A:)
meaipvkqfvkhigelysnnqhgfsedfeevqrctadmnitaehsnhpenkhknryinil
aydhsrvklrplpgskhsdyinanyvdgynkakayiatqgplkstfedfwrmiweqntgi
ivmitnlvekgrrkcdqywptenseeygniivtlkstkihacytvrrfsirntkqnervv
iqyhytqwpdmgvpeyalpvltfvrrssaarmpetgpvlvhcsagvgrtgtyividsmlq
qikdkstvnvlgflkhirtqrnylvqteeqyifihdalleailgk