PDB entry 3qcj

View 3qcj on RCSB PDB site
Description: Human receptor protein tyrosine phosphatase gamma, domain 1, in complex with 5-[({3-[(3,4-dichlorobenzyl)sulfanyl]thiophen-2-yl}carbonyl)sulfamoyl]-2-methoxybenzoic acid
Class: hydrolase/hydrolase inhibitor
Keywords: TYROSINE RECEPTOR PHOSPHATASE, TWISTED MIXED BETA-SHEETS FLANKED BY {ALPHA}-HELICES, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on 2011-01-16, released 2011-12-28
The last revision prior to the SCOPe 2.05 freeze date was dated 2011-12-28, with a file datestamp of 2011-12-23.
Experiment type: XRAY
Resolution: 2.26 Å
R-factor: 0.215
AEROSPACI score: 0.38 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Receptor-type tyrosine-protein phosphatase gamma
    Species: Homo sapiens [TaxId:9606]
    Gene: PTPG, PTPRG
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.05: d3qcja_
  • Heterogens: NX4, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3qcjA (A:)
    gshmgsmeaipvkqfvkhigelysnnqhgfsedfeevqrctadmnitaehsnhpenkhkn
    ryinilaydhsrvklrplpgkdskhsdyinanyvdgynkakayiatqgplkstfedfwrm
    iweqntgiivmitnlvekgrrkcdqywptenseeygniivtlkstkihacytvrrfsirn
    tkvkkgqkgnpkgrqnervviqyhytqwpdmgvpeyalpvltfvrrssaarmpetgpvlv
    hcsagvgrtgtyividsmlqqikdkstvnvlgflkhirtqrnylvqteeqyifihdalle
    ailgketevs
    

    Sequence, based on observed residues (ATOM records): (download)
    >3qcjA (A:)
    meaipvkqfvkhigelysnnqhgfsedfeevqrctadmnitaehsnhpenkhknryinil
    aydhsrvklrplpgskhsdyinanyvdgynkakayiatqgplkstfedfwrmiweqntgi
    ivmitnlvekgrrkcdqywptenseeygniivtlkstkihacytvrrfsirntkqnervv
    iqyhytqwpdmgvpeyalpvltfvrrssaarmpetgpvlvhcsagvgrtgtyividsmlq
    qikdkstvnvlgflkhirtqrnylvqteeqyifihdalleailgk