PDB entry 3q3s
View 3q3s on RCSB PDB site
Description: EthR from Mycobacterium tuberculosis in complex with compound BDM5683
Class: transcription repressor/inhibitor
Keywords: Antitubercular Agents, DNA-Binding Protein, Repressor Proteins, Tuberculosis, TRANSCRIPTION REPRESSOR-INHIBITOR complex
Deposited on
2010-12-22, released
2012-01-18
The last revision prior to the SCOPe 2.08 freeze date was dated
2012-01-18, with a file datestamp of
2012-01-13.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.191
AEROSPACI score: 0.47
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: HTH-type transcriptional regulator EthR
Species: Mycobacterium tuberculosis [TaxId:1773]
Gene: ethR, etaR, MT3970, Rv3855
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3q3sa1, d3q3sa2 - Heterogens: O8B, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3q3sA (A:)
mgsshhhhhhssglvprgshmttsaasqaslprgrrtarpsgddrelailataenlledr
pladisvddlakgagisrptfyfyfpskeavlltlldrvvnqadmalqtlaenpadtdre
nmwrtginvffetfgshkavtragqaaratsvevaelwstfmqkwiaytaavidaerdrg
aaprtlpahelatalnlmnertlfasfageqpsvpearvldtlvhiwvtsiygenr
Sequence, based on observed residues (ATOM records): (download)
>3q3sA (A:)
gddrelailataenlledrpladisvddlakgagisrptfyfyfpskeavlltlldrvvn
qadmalqtlaenpadtdrenmwrtginvffetfgshkavtragqaaratsvevaelwstf
mqkwiaytaavidaerdrgaaprtlpahelatalnlmnertlfasfageqpsvpearvld
tlvhiwvtsiygen