PDB entry 3q3s

View 3q3s on RCSB PDB site
Description: EthR from Mycobacterium tuberculosis in complex with compound BDM5683
Class: transcription repressor/inhibitor
Keywords: Antitubercular Agents, DNA-Binding Protein, Repressor Proteins, Tuberculosis, TRANSCRIPTION REPRESSOR-INHIBITOR complex
Deposited on 2010-12-22, released 2012-01-18
The last revision prior to the SCOPe 2.08 freeze date was dated 2012-01-18, with a file datestamp of 2012-01-13.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.191
AEROSPACI score: 0.47 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: HTH-type transcriptional regulator EthR
    Species: Mycobacterium tuberculosis [TaxId:1773]
    Gene: ethR, etaR, MT3970, Rv3855
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d3q3sa1, d3q3sa2
  • Heterogens: O8B, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3q3sA (A:)
    mgsshhhhhhssglvprgshmttsaasqaslprgrrtarpsgddrelailataenlledr
    pladisvddlakgagisrptfyfyfpskeavlltlldrvvnqadmalqtlaenpadtdre
    nmwrtginvffetfgshkavtragqaaratsvevaelwstfmqkwiaytaavidaerdrg
    aaprtlpahelatalnlmnertlfasfageqpsvpearvldtlvhiwvtsiygenr
    

    Sequence, based on observed residues (ATOM records): (download)
    >3q3sA (A:)
    gddrelailataenlledrpladisvddlakgagisrptfyfyfpskeavlltlldrvvn
    qadmalqtlaenpadtdrenmwrtginvffetfgshkavtragqaaratsvevaelwstf
    mqkwiaytaavidaerdrgaaprtlpahelatalnlmnertlfasfageqpsvpearvld
    tlvhiwvtsiygen