PDB entry 3pze
View 3pze on RCSB PDB site
Description: JNK1 in complex with inhibitor
Class: transferase/transferase inhibitor
Keywords: kinase JNK1, inhibitor, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-12-14, released
2011-12-14
The last revision prior to the SCOPe 2.06 freeze date was dated
2012-06-27, with a file datestamp of
2012-06-22.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.206
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 8
Species: Homo sapiens [TaxId:9606]
Gene: MAPK8, JNK1, PRKM8, SAPK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3pzea_ - Heterogens: SO4, CFK, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3pzeA (A:)
dnnfysveigdstftvlkryqnlkpigsgaqgivcaaydailernvaikklsrpfqnqth
akrayrelvlmkcvnhkniigllnvftpqksleefqdvyivmelmdanlcqviqmeldhe
rmsyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartagtsfmmtpyv
vtryyrapevilgmgykenvdlwsvgcimgemvchkilfpgrdyidqwnkvieqlgtpcp
efmkklqptvrtyvenrpkyagysfeklfpdvlfpadsehnklkasqardllskmlvida
skrisvdealqhpyinvwydpseaeapppkipdkqlderehtieewkeliykevmdle
Sequence, based on observed residues (ATOM records): (download)
>3pzeA (A:)
dnnfysveigdstftvlkryqnlkpigsgaqgivcaaydailernvaikklsrpfqnqth
akrayrelvlmkcvnhkniigllnvftpqksleefqdvyivmelmdanlcqviqmeldhe
rmsyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglsfmmtvtryyrape
vilgmgykenvdlwsvgcimgemvchkilfpgrdyidqwnkvieqlgtpcpefmkklqpt
vrtyvenrpkyagysfeklfpdvlfpadsehnklkasqardllskmlvidaskrisvdea
lqhpyinvwydpseaeapppkipdkqlderehtieewkeliykevmd