PDB entry 3pyy
View 3pyy on RCSB PDB site
Description: Discovery and Characterization of a Cell-Permeable, Small-molecule c-Abl Kinase Activator that Binds to the Myristoyl Binding Site
Class: transferase
Keywords: Tyrosine kinase, Transferase
Deposited on
2010-12-13, released
2011-03-09
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-01-24, with a file datestamp of
2018-01-19.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: N/A
AEROSPACI score: 0.36
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: V-abl Abelson murine leukemia viral oncogene homolog 1 isoform b variant
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3pyya1, d3pyya2 - Chain 'B':
Compound: V-abl Abelson murine leukemia viral oncogene homolog 1 isoform b variant
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3pyyb1, d3pyyb2 - Heterogens: SO4, STI, 3YY, 2PE, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3pyyA (A:)
mhhhhhhenlyfqgspnydkwemertditmkhklgggqygevyegvwkkysltvavktlk
edtmeveeflkeaavmkeikhpnlvqllgvctreppfyiitefmtygnlldylrecnrqe
vnavvllymatqissameylekknfihrdlaarnclvgenhlvkvadfglsrlmtgdtyt
ahagakfpikwtapeslaynkfsiksdvwafgvllweiatygmspypgidlsqvyellek
dyrmerpegcpekvyelmracwqwnpsdrpsfaeihqafetmfqessisdevekelgk
Sequence, based on observed residues (ATOM records): (download)
>3pyyA (A:)
ydkwemertditmkhklgggqygevyegvwkkysltvavktlkeveeflkeaavmkeikh
pnlvqllgvctreppfyiitefmtygnlldylrecnrqevnavvllymatqissameyle
kknfihrdlaarnclvgenhlvkvadfglsrlmtgdtytahagakfpikwtapeslaynk
fsiksdvwafgvllweiatygmspypgidlsqvyellekdyrmerpegcpekvyelmrac
wqwnpsdrpsfaeihqafetmfqes
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3pyyB (B:)
mhhhhhhenlyfqgspnydkwemertditmkhklgggqygevyegvwkkysltvavktlk
edtmeveeflkeaavmkeikhpnlvqllgvctreppfyiitefmtygnlldylrecnrqe
vnavvllymatqissameylekknfihrdlaarnclvgenhlvkvadfglsrlmtgdtyt
ahagakfpikwtapeslaynkfsiksdvwafgvllweiatygmspypgidlsqvyellek
dyrmerpegcpekvyelmracwqwnpsdrpsfaeihqafetmfqessisdevekelgk
Sequence, based on observed residues (ATOM records): (download)
>3pyyB (B:)
dkwemertditmkhklgggqygevyegvwkkysltvavktlveeflkeaavmkeikhpnl
vqllgvctreppfyiitefmtygnlldylrecnrqevnavvllymatqissameylekkn
fihrdlaarnclvgenhlvkvadfgakfpikwtapeslaynkfsiksdvwafgvllweia
tygmspypgidlsqvyellekdyrmerpegcpekvyelmracwqwnpsdrpsfaeihqaf
etmfqessisdevekel