PDB entry 3pvu
View 3pvu on RCSB PDB site
Description: Bovine GRK2 in complex with Gbetagamma subunits and a selective kinase inhibitor (CMPD101)
Class: transferase/signaling protein/inhibitor
Keywords: Transferase, Serine/threonine-protein kinase, ATP-binding, Inhibitor, Membrane, TRANSFERASE-SIGNALING PROTEIN-INHIBITOR complex
Deposited on
2010-12-07, released
2011-06-01
The last revision prior to the SCOPe 2.02 freeze date was dated
2011-07-27, with a file datestamp of
2011-07-22.
Experiment type: XRAY
Resolution: 2.48 Å
R-factor: 0.229
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Beta-adrenergic receptor kinase 1
Species: Bos taurus [TaxId:9913]
Gene: ADRBK1, GRK2
Database cross-references and differences (RAF-indexed):
- Chain 'B':
Compound: Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1
Species: Bos taurus [TaxId:9913]
Gene: GNB1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d3pvub_ - Chain 'G':
Compound: Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2
Species: Bos taurus [TaxId:9913]
Gene: GNG2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d3pvug_ - Heterogens: QRW, HOH
PDB Chain Sequences:
- Chain 'A':
No sequence available.
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3pvuB (B:)
mseldqlrqeaeqlknqirdarkacadatlsqitnnidpvgriqmrtrrtlrghlakiya
mhwgtdsrllvsasqdgkliiwdsyttnkvhaiplrsswvmtcayapsgnyvacggldni
csiynlktregnvrvsrelaghtgylsccrflddnqivtssgdttcalwdietgqqtttf
tghtgdvmslslapdtrlfvsgacdasaklwdvregmcrqtftghesdinaicffpngna
fatgsddatcrlfdlradqelmtyshdniicgitsvsfsksgrlllagyddfncnvwdal
kadragvlaghdnrvsclgvtddgmavatgswdsflkiwn
Sequence, based on observed residues (ATOM records): (download)
>3pvuB (B:)
seldqlrqeaeqlknqirdarkacadatlsqitnnidpvgriqmrtrrtlrghlakiyam
hwgtdsrllvsasqdgkliiwdsyttnkvhaiplrsswvmtcayapsgnyvacggldnic
siynlktregnvrvsrelaghtgylsccrflddnqivtssgdttcalwdietgqqtttft
ghtgdvmslslapdtrlfvsgacdasaklwdvregmcrqtftghesdinaicffpngnaf
atgsddatcrlfdlradqelmtyshdniicgitsvsfsksgrlllagyddfncnvwdalk
adragvlaghdnrvsclgvtddgmavatgswdsflkiwn
- Chain 'G':
Sequence, based on SEQRES records: (download)
>3pvuG (G:)
hhhhhhmasnntasiaqarklveqlkmeanidrikvskaaadlmayceahakedplltpv
pasenpfrekkffc
Sequence, based on observed residues (ATOM records): (download)
>3pvuG (G:)
siaqarklveqlkmeanidrikvskaaadlmayceahakedplltpvpasenpfrekkff
c