PDB entry 3pp1
View 3pp1 on RCSB PDB site
Description: Crystal Structure of the Human Mitogen-activated protein kinase kinase 1 (MEK 1) in complex with ligand and MgATP
Class: transferase/transferase inhibitor
Keywords: Kinase domain, Kinase, ATP binding, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-11-23, released
2011-02-23
The last revision prior to the SCOPe 2.02 freeze date was dated
2011-03-09, with a file datestamp of
2011-03-04.
Experiment type: XRAY
Resolution: 2.7 Å
R-factor: 0.184
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dual specificity mitogen-activated protein kinase kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: MAP2K1, Mapk/erk kinase 1, MEK1, PRKMK1
Database cross-references and differences (RAF-indexed):
- Uniprot Q02750 (1-321)
- initiating methionine (0)
Domains in SCOPe 2.02: d3pp1a_ - Heterogens: ATP, MG, IZG, ACT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3pp1A (A:)
melkdddfekiselgagnggvvfkvshkpsglvmarklihleikpairnqiirelqvlhe
cnspyivgfygafysdgeisicmehmdggsldqvlkkagripeqilgkvsiavikgltyl
rekhkimhrdvkpsnilvnsrgeiklcdfgvsgqlidsmansfvgtrsymsperlqgthy
svqsdiwsmglslvemavgrypipppdakelelmfgcqvegdaaetpprprtpgrplssy
gmdsrppmaifelldyivnepppklpsgvfslefqdfvnkcliknpaeradlkqlmvhaf
ikrsdaeevdfagwlcstiglnhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3pp1A (A:)
melkdddfekiselgagnggvvfkvshkpsglvmarklihleikpairnqiirelqvlhe
cnspyivgfygafysdgeisicmehmdggsldqvlkkagripeqilgkvsiavikgltyl
rekhkimhrdvkpsnilvnsrgeiklcdfgvsgqlidsmansfvgtrsymsperlqgthy
svqsdiwsmglslvemavgrypipppdakelelmfpmaifelldyivnepppklpsgvfs
lefqdfvnkcliknpaeradlkqlmvhafikrsdaeevdfagwlcstigln