PDB entry 3poz
View 3poz on RCSB PDB site
Description: EGFR Kinase domain complexed with tak-285
Class: transferase/transferase inhibitor
Keywords: KINASE DOMAIN, ANTI-ONCOGENE, ATP-BINDING, CELL CYCLE, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, RECEPTOR, SECRETED, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-11-23, released
2011-03-30
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-06-15, with a file datestamp of
2011-06-10.
Experiment type: XRAY
Resolution: 1.5 Å
R-factor: 0.22
AEROSPACI score: 0.6
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3poza_ - Heterogens: SO4, 03P, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3pozA (A:)
geapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreatspka
nkeildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqyll
nwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyhaeggk
vpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerlpq
ppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpsptds
nfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>3pozA (A:)
qallrilketefkkikvlgsgafgtvykglwipvkipvaikelankeildeayvmasvdn
phvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqyllnwcvqiakgmnyledr
rlvhrdlaarnvlvktpqhvkitdfglakllgaeekkvpikwmalesilhriythqsdvw
sygvtvwelmtfgskpydgipaseissilekgerlpqppictidvymimvkcwmidadsr
pkfreliiefskmardpqrylviqgdermhlpsptdsnfyralmdvvdadeyl