PDB entry 3pb1
View 3pb1 on RCSB PDB site
Description: Crystal Structure of a Michaelis Complex between Plasminogen Activator Inhibitor-1 and Urokinase-type Plasminogen Activator
Class: hydrolase Inhibitor/Hydrolase
Keywords: PAI-1, uPA, Michaelis complex, Structural Genomics, Structure 2 Function Project, S2F, hydrolase Inhibitor-Hydrolase complex
Deposited on
2010-10-20, released
2010-12-29
The last revision prior to the SCOPe 2.07 freeze date was dated
2011-03-09, with a file datestamp of
2011-03-04.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: 0.223
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'E':
Compound: Plasminogen activator, urokinase
Species: Homo sapiens [TaxId:9606]
Gene: PLAU, RP11-417O11.1-002
Database cross-references and differences (RAF-indexed):
- Uniprot Q5SWW8 (0-End)
- conflict (120)
- conflict (143)
- engineered mutation (197)
Domains in SCOPe 2.07: d3pb1e_ - Chain 'I':
Compound: Plasminogen activator inhibitor 1
Species: Homo sapiens [TaxId:9606]
Gene: SERPINE1, PAI1, PLANH1
Database cross-references and differences (RAF-indexed):
- Uniprot P05121 (Start-378)
- engineered mutation (149)
- engineered mutation (153)
- conflict (157)
- engineered mutation (318)
- engineered mutation (353)
Domains in SCOPe 2.07: d3pb1i_ - Heterogens: SO4, HOH
PDB Chain Sequences:
- Chain 'E':
Sequence, based on SEQRES records: (download)
>3pb1E (E:)
iiggefttienqpwfaaiyrrhrggsvtyvcggslispcwvisathcfidypkkedyivy
lgrsrlnsntqgemkfevenlilhkdysadtlahhndiallkirskegrcaqpsrtiqti
alpsmyndpqfgtsceitgfgkeqstdylypeqlkmtvvklishrecqqphyygsevttk
mlcaadpqwktdscqgdaggplvcslqgrmtltgivswgrgcalkdkpgvytrvshflpw
irshtkeenglal
Sequence, based on observed residues (ATOM records): (download)
>3pb1E (E:)
iiggefttienqpwfaaiyrrhrggsvtyvcggslispcwvisathcfidypkkedyivy
lgrsrlnsntqgemkfevenlilhkdysadtlahhndiallkirskegrcaqpsrtiqti
alpsmyndpqfgtsceitgfgkeqstdylypeqlkmtvvklishrecqqphyygsevttk
mlcaadpqwktdscqgdaggplvcslqgrmtltgivswgrgcalkdkpgvytrvshflpw
irshtke
- Chain 'I':
Sequence, based on SEQRES records: (download)
>3pb1I (I:)
vhhppsyvahlasdfgvrvfqqvaqaskdrnvvfspygvasvlamlqlttggetqqqiqa
amgfkiddkgmapalrhlykelmgpwnkdeisttdaifvqrdlklvqgfmphffrlfrst
vkqvdfseverarfiindwvkthtkgmishllgtgavqqltrlvlvnalyfngqwktpfp
dssthrrlfhksdgstvsvpmmaqtnkfnytefttpdghyydilelpyhgdtlsmfiaap
yekevplsaltnilsaqlishwkgnmtrlprllvlpkfsletevdlrkplenlgmtdmfr
qfqadftslsdqeplhvalalqkvkievnesgtvassstavivsarmapeeiiidrpflf
vvrhnptgtvlfmgqvmep
Sequence, based on observed residues (ATOM records): (download)
>3pb1I (I:)
psyvahlasdfgvrvfqqvaqaskdrnvvfspygvasvlamlqlttggetqqqiqaamgf
kiddkgmapalrhlykelmgpwnkdeisttdaifvqrdlklvqgfmphffrlfrstvkqv
dfseverarfiindwvkthtkgmishllgtgavqqltrlvlvnalyfngqwktpfpdsst
hrrlfhksdgstvsvpmmaqtnkfnytefttpdghyydilelpyhgdtlsmfiaapyeke
vplsaltnilsaqlishwkgnmtrlprllvlpkfsletevdlrkplenlgmtdmfrqfqa
dftslsdqeplhvalalqkvkievnesgtvassstavivsarmapeeiiidrpflfvvrh
nptgtvlfmgqvmep