PDB entry 3pa4
View 3pa4 on RCSB PDB site
Description: X-ray crystal structure of compound 2a bound to human CHK1 kinase domain
Class: transferase/transferase inhibitor
Keywords: kinase, phosphatase, transferase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-10-18, released
2010-12-08
The last revision prior to the SCOPe 2.05 freeze date was dated
2010-12-08, with a file datestamp of
2010-12-03.
Experiment type: XRAY
Resolution: 1.59 Å
R-factor: 0.225
AEROSPACI score: 0.53
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3pa4a_ - Heterogens: C72, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3pa4A (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkm
lnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvyl
hgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkr
refhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplal
lhkilvenpsaritipdikkdrwynkplkkgak
Sequence, based on observed residues (ATOM records): (download)
>3pa4A (A:)
vedwdlvqtlgegaygevqlavnrvteeavavkivdmnikkeicinkmlnhenvvkfygh
rregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithrdikp
enlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepvdvws
cgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilvenpsar
itipdikkdrwynkplkkg