PDB entry 3p88
View 3p88 on RCSB PDB site
Description: FXR bound to isoquinolinecarboxylic acid
Class: transcription/inhibitor
Keywords: nuclear recptor FXR, TRANSCRIPTION-INHIBITOR complex
Deposited on
2010-10-13, released
2011-08-31
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-11-08, with a file datestamp of
2017-11-03.
Experiment type: XRAY
Resolution: 2.95 Å
R-factor: N/A
AEROSPACI score: 0.15
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Farnesoid X receptor
Species: Homo sapiens [TaxId:9606]
Gene: hCG_20893, NR1H4
Database cross-references and differences (RAF-indexed):
- Uniprot B6ZGS9 (0-228)
- conflict (41)
- engineered mutation (188)
- engineered mutation (222)
Domains in SCOPe 2.08: d3p88a_ - Chain 'B':
Compound: Nuclear receptor coactivator 1
Species: Homo sapiens [TaxId:9606]
Gene: BHLHE74, NCOA1, SRC1
Database cross-references and differences (RAF-indexed):
- Heterogens: P88, SO4, HOH