PDB entry 3oct
View 3oct on RCSB PDB site
Description: Crystal structure of bruton's tyrosine kinase mutant V555R in complex with dasatinib
Class: transferase/transferase inhibitor
Keywords: tyrosine kinase, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-08-10, released
2010-11-03
The last revision prior to the SCOPe 2.02 freeze date was dated
2010-11-17, with a file datestamp of
2010-11-12.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: 0.199
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Tyrosine-protein kinase BTK
Species: Homo sapiens [TaxId:9606]
Gene: BTK, AGMX1, ATK, BPK
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d3octa_ - Heterogens: 1N1, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3octA (A:)
ggsweidpkdltflkelgtgqfgvvkygkwrgqydvaikmikegsmsedefieeakvmmn
lsheklvqlygvctkqrpifiiteymangcllnylremrhrfqtqqllemckdvceamey
leskqflhrdlaarnclvndqgvvkvsdfglsryvlddeytssrgskfpvrwsppevlmy
skfssksdiwafgvlmweiyslgkmpyerftnsetaehiaqglrlyrphlasekvytimy
scwhekaderptfkillsnildvmd
Sequence, based on observed residues (ATOM records): (download)
>3octA (A:)
sweidpkdltflkelgqfgvvkygkwrgqydvaikmikmsedefieeakvmmnlsheklv
qlygvctkqrpifiiteymangcllnylremrhrfqtqqllemckdvceameyleskqfl
hrdlaarnclvndqgvvkvsdfglsrfpvrwsppevlmyskfssksdiwafgvlmweiys
lgkmpyerftnsetaehiaqglrlyrphlasekvytimyscwhekaderptfkillsnil
dvmd