PDB entry 3o2f

View 3o2f on RCSB PDB site
Description: Structure of the N-domain of GRP94 bound to the HSP90 inhibitor PU-H54
Class: chaperone/inhibitor
Keywords: Hsp90 Heat-shock Proteins, chaperone-inhibitor complex
Deposited on 2010-07-22, released 2011-10-05
The last revision prior to the SCOPe 2.07 freeze date was dated 2017-08-23, with a file datestamp of 2017-08-18.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Endoplasmin
    Species: Canis lupus familiaris [TaxId:9615]
    Gene: GRP94, HSP90B1, TRA1
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d3o2fa_
  • Chain 'B':
    Compound: Endoplasmin
    Species: Canis lupus familiaris [TaxId:9615]
    Gene: GRP94, HSP90B1, TRA1
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d3o2fb_
  • Heterogens: P54, IPA, GOL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3o2fA (A:)
    gshmlreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltden
    alagneeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqed
    gqstseligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrg
    ttitlvlkeeasdyleldtiknlvkkysqfinfpiyvwssktggggktvwdwelmn
    

    Sequence, based on observed residues (ATOM records): (download)
    >3o2fA (A:)
    lreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltdenalag
    neeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqedgqst
    seligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrgttit
    lvlkeeasdyleldtiknlvkkysqfinfpiyvwssktktvwdwelmn
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >3o2fB (B:)
    gshmlreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltden
    alagneeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqed
    gqstseligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrg
    ttitlvlkeeasdyleldtiknlvkkysqfinfpiyvwssktggggktvwdwelmn
    

    Sequence, based on observed residues (ATOM records): (download)
    >3o2fB (B:)
    ekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltdenalagneelt
    vkikcdkeknllhvtdtgvgmtreelvknlgtiakseflmteaqedgqstseligqfgvg
    fysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrgttitlvlkeeasdy
    leldtiknlvkkysqfinfpiyvwssktktvwdwelmn