PDB entry 3nw7
View 3nw7 on RCSB PDB site
Description: Crystal structure of insulin-like growth factor 1 receptor (IGF-1R-WT) complex with a carbon-linked proline isostere inhibitor (34)
Class: transferase
Keywords: hormone/growth factor, igf-1r, kinase domain, transferase
Deposited on
2010-07-09, released
2010-07-28
The last revision prior to the SCOPe 2.08 freeze date was dated
2010-09-08, with a file datestamp of
2010-09-03.
Experiment type: XRAY
Resolution: 2.11 Å
R-factor: 0.168
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: insulin-like growth factor 1 receptor
Species: Homo sapiens [TaxId:9606]
Gene: IGF1R
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3nw7a_ - Heterogens: LGV, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3nw7A (A:)
mvsaadvyvpdewevarekitmsrelgqgsfgmvyegvakgvvkdepetrvaiktvneaa
smrerieflneasvmkefnchhvvrllgvvsqgqptlvimelmtrgdlksylrslrpeme
nnpvlappslskmiqmageiadgmaylnankfvhrdlaarncmvaedftvkigdfgmtrd
iyetdyyrkggkgllpvrwmspeslkdgvfttysdvwsfgvvlweiatlaeqpyqglsne
qvlrfvmegglldkpdncpdmlfelmrmcwqynpkmrpsfleiissikeemepgfrevsf
yyseenk
Sequence, based on observed residues (ATOM records): (download)
>3nw7A (A:)
yvpdewevarekitmsrelgqgsfgmvyegvakgvvkdepetrvaiktvneaasmrerie
flneasvmkefnchhvvrllgvvsqgqptlvimelmtrgdlksylrslrpemennpvlap
pslskmiqmageiadgmaylnankfvhrdlaarncmvaedftvkigdfgmtrdiyetdyy
rkgllpvrwmspeslkdgvfttysdvwsfgvvlweiatlaeqpyqglsneqvlrfvmegg
lldkpdncpdmlfelmrmcwqynpkmrpsfleiissikeemepgfrevsfyyseenk