PDB entry 3nrm
View 3nrm on RCSB PDB site
Description: Imidazo[1,2-a]pyrazine-based Aurora Kinase Inhibitors
Class: transferase
Keywords: kinase, cell cycle, inhibitor, transferase
Deposited on
2010-06-30, released
2010-08-18
The last revision prior to the SCOPe 2.06 freeze date was dated
2010-09-22, with a file datestamp of
2010-09-17.
Experiment type: XRAY
Resolution: 3.05 Å
R-factor: 0.223
AEROSPACI score: 0.21
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine-protein kinase 6
Species: Homo sapiens [TaxId:9606]
Gene: AURKA, AIK, ARK1, AURA, BTAK, STK15, STK6
Database cross-references and differences (RAF-indexed):
- Uniprot O14965 (5-End)
- engineered mutation (166-167)
Domains in SCOPe 2.06: d3nrma_ - Heterogens: NRM
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3nrmA (A:)
gamgsrqwaledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrr
eveiqshlrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitel
analsychskrvihrdikpenlllgsagelkiadfgwsvhapssrraalcgtldylppem
iegrmhdekvdlwslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardli
srllkhnpsqrpmlrevlehpwitansskpsncqnkesaskqs
Sequence, based on observed residues (ATOM records): (download)
>3nrmA (A:)
rqwaledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrreveiq
shlrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitelanals
ychskrvihrdikpenlllgsagelkiadfgwsvhapssrraalcgtldylppemiegrm
hdekvdlwslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardlisrllk
hnpsqrpmlrevlehpwitanss