PDB entry 3n6k
View 3n6k on RCSB PDB site
Description: Human FPPS complex with NOV_823
Class: transferase/transferase inhibitor
Keywords: BISPHOSPHONATE; FRAGMENT-BASED SCREENING; TRANSFERASE; ISOPRENE BIOSYNTHESIS; CHOLESTEROL BIOSYNTHESIS, RANSFERASE-TRANSFERASE INHIBITOR complex, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-05-26, released
2010-08-18
The last revision prior to the SCOPe 2.06 freeze date was dated
2010-09-01, with a file datestamp of
2010-08-27.
Experiment type: XRAY
Resolution: 2.25 Å
R-factor: 0.265
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'F':
Compound: farnesyl pyrophosphate synthase
Species: Homo sapiens [TaxId:9606]
Gene: FDPS, FPS, KIAA1293
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3n6kf_ - Heterogens: BFH, PO4, HOH
PDB Chain Sequences:
- Chain 'F':
Sequence, based on SEQRES records: (download)
>3n6kF (F:)
gpnsdvyaqekqdfvqhfsqivrvltedemghpeigdaiarlkevleynaiggkynrglt
vvvafrelveprkqdadslqrawtvgwcvellqafflvaddimdssltrrgqicwyqkpg
vgldaindanlleaciyrllklycreqpyylnlielflqssyqteigqtldlltapqgnv
dlvrftekryksivkyktafysfylpiaaamymagidgekehanakkillemgeffqiqd
dyldlfgdpsvtgkigtdiqdnkcswlvvqclqratpeqyqilkenygqkeaekvarvka
lyeeldlpavflqyeedsyshimalieqyaaplppavflglarkiykrrk
Sequence, based on observed residues (ATOM records): (download)
>3n6kF (F:)
yaqekqdfvqhfsqivrvltedemghpeigdaiarlkevleynaiggkynrgltvvvafr
elveprkqdadslqrawtvgwcvellqafflvaddimdssltrrgqicwyqkpgvgldai
ndanlleaciyrllklycreqpyylnlielflqssyqteigqtldlltapqgnvdlvrft
ekryksivkyktafysfylpiaaamymagidgekehanakkillemgeffqiqddyldlf
gdpsvtgkigtdiqdnkcswlvvqclqratpeqyqilkenygqkeaekvarvkalyeeld
lpavflqyeedsyshimalieqyaaplppavflglarkiyk