PDB entry 3mw1
View 3mw1 on RCSB PDB site
Description: p38 kinase Crystal structure in complex with small molecule inhibitor
Class: TRANSFERASE/TRANSFERASE inhibitor
Keywords: p38 MAP KINASE, TRANSFERASE, INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE inhibitor complex
Deposited on
2010-05-05, released
2011-04-27
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-12-07, with a file datestamp of
2011-12-02.
Experiment type: XRAY
Resolution: 2.8 Å
R-factor: 0.259
AEROSPACI score: 0.21
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: Mapk14
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3mw1a_ - Heterogens: MIH, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3mw1A (A:)
sqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqs
iihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqk
ltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemtg
yvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgt
pgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaq
alahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3mw1A (A:)
erptfyrqelnktiwevperyqnlspvgsvcaafdtktglrvavkklsrpfqsiihakrt
yrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltddhvq
fliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglatddemtgyvatrwyra
peimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkki
ssesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaq
yhdpddepvadpydqsfesrdllidewksltydevisfvppp