PDB entry 3miy
View 3miy on RCSB PDB site
Description: X-ray crystal structure of ITK complexed with sunitinib
Class: Transferase
Keywords: helix C-in, Transferase
Deposited on
2010-04-12, released
2010-06-30
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-10-05, with a file datestamp of
2011-09-30.
Experiment type: XRAY
Resolution: 1.67 Å
R-factor: 0.208
AEROSPACI score: 0.54
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Tyrosine-protein kinase ITK/TSK
Species: Homo sapiens [TaxId:9606]
Gene: ITK, EMT, LYK
Database cross-references and differences (RAF-indexed):
- Uniprot Q08881 (2-End)
- expression tag (0-1)
- engineered (122)
- engineered (259)
- engineered (262)
Domains in SCOPe 2.06: d3miya1, d3miya2 - Chain 'B':
Compound: Tyrosine-protein kinase ITK/TSK
Species: Homo sapiens [TaxId:9606]
Gene: ITK, EMT, LYK
Database cross-references and differences (RAF-indexed):
- Uniprot Q08881 (2-End)
- expression tag (0-1)
- engineered (122)
- engineered (259)
- engineered (262)
Domains in SCOPe 2.06: d3miyb1, d3miyb2 - Heterogens: B49, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3miyA (A:)
gsvidpseltfvqeigsgqfglvhlgywlnkdkvaiktiregamseedfieeaevmmkls
hpklvqlygvcleqapiclvfefmehgclsdylrtqrglfaaetllgmcldvcegmayle
easvihrdlaarnclvgenqvikvsdfgmtrfvlddqytsstgtkfpvkwaspevfsfsr
yssksdvwsfgvlmwevfsegkipyenrsnsevvedistgfrlykprlasthvyqimnhc
wkerpedrpafsrllrqlaaiaasgl
Sequence, based on observed residues (ATOM records): (download)
>3miyA (A:)
gsvidpseltfvqeigsgglvhlgywlnkdkvaiktiseedfieeaevmmklshpklvql
ygvcleqapiclvfefmehgclsdylrtqrglfaaetllgmcldvcegmayleeasvihr
dlaarnclvgenqvikvsdfpvkwaspevfsfsryssksdvwsfgvlmwevfsegkipye
nrsnsevvedistgfrlykprlasthvyqimnhcwkerpedrpafsrllrqlaaiaasg
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3miyB (B:)
gsvidpseltfvqeigsgqfglvhlgywlnkdkvaiktiregamseedfieeaevmmkls
hpklvqlygvcleqapiclvfefmehgclsdylrtqrglfaaetllgmcldvcegmayle
easvihrdlaarnclvgenqvikvsdfgmtrfvlddqytsstgtkfpvkwaspevfsfsr
yssksdvwsfgvlmwevfsegkipyenrsnsevvedistgfrlykprlasthvyqimnhc
wkerpedrpafsrllrqlaaiaasgl
Sequence, based on observed residues (ATOM records): (download)
>3miyB (B:)
gsvidpseltfvqeigsgglvhlgywlnkdkvaiktiseedfieeaevmmklshpklvql
ygvcleqapiclvfefmehgclsdylrtqrglfaaetllgmcldvcegmayleeasvihr
dlaarnclvgenqvikvsdfgpvkwaspevfsfsryssksdvwsfgvlmwevfsegkipy
enrsnsevvedistgfrlykprlasthvyqimnhcwkerpedrpafsrllrqlaaiaasg