PDB entry 3l8p
View 3l8p on RCSB PDB site
Description: Crystal structure of cytoplasmic kinase domain of Tie2 complexed with inhibitor CEP11207
Class: transferase
Keywords: receptor tyrosine kinase, cytoplasmic kinase domain, Tie2, inhibitor CEP11207, ATP-binding, Disease mutation, Glycoprotein, Kinase, Membrane, Nucleotide-binding, Phosphoprotein, Receptor, Transferase, Tyrosine-protein kinase
Deposited on
2010-01-03, released
2010-10-06
The last revision prior to the SCOPe 2.05 freeze date was dated
2010-10-06, with a file datestamp of
2010-10-01.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.238
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Angiopoietin-1 receptor
Species: Homo sapiens [TaxId:9606]
Gene: TEK, TIE2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3l8pa_ - Heterogens: 0CE, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3l8pA (A:)
knnpdptiypvldwndikfqdvigegnfgqvlkarikkdglrmdaaikrmkeyaskddhr
dfagelevlcklghhpniinllgacehrgylylaieyaphgnlldflrksrvletdpafa
ianstastlssqqllhfaadvargmdylsqkqfihrdlaarnilvgenyvakiadfglsr
gqevyvkktmgrlpvrwmaieslnysvyttnsdvwsygvllweivslggtpycgmtcael
yeklpqgyrlekplncddevydlmrqcwrekpyerpsfaqilvslnrmleerktyvnttl
yekftyagidcsaeeaa
Sequence, based on observed residues (ATOM records): (download)
>3l8pA (A:)
tiypvldwndikfqdvigegnfgqvlkarikkdglrmdaaikrmfagelevlcklghhpn
iinllgacehrgylylaieyaphgnlldflrksrvletdpafaianstastlssqqllhf
aadvargmdylsqkqfihrdlaarnilvgenyvakiadfglsrgqevyvkkpvrwmaies
lnysvyttnsdvwsygvllweivslggtpycgmtcaelyeklpqgyrlekplncddevyd
lmrqcwrekpyerpsfaqilvslnrmleerktyvnttlyekftyagidcsae