PDB entry 3krl
View 3krl on RCSB PDB site
Description: cFMS Tyrosine kinase in complex with 5-Cyano-furan-2-carboxylic acid [4-(4-methyl-piperazin-1-yl)-2-piperidin-1-yl-phenyl]-amide
Class: transferase/transferase inhibitor
Keywords: Kinase, inhibitor, chimera, ATP-binding, Disulfide bond, Glycoprotein, Immunoglobulin domain, Membrane, Nucleotide-binding, Phosphoprotein, Proto-oncogene, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2009-11-18, released
2010-12-01
The last revision prior to the SCOPe 2.04 freeze date was dated
2011-12-14, with a file datestamp of
2011-12-09.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.212
AEROSPACI score: 0.2
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Macrophage colony-stimulating factor 1 receptor, Basic fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: CSF1R, FGFR1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d3krla_ - Heterogens: KRL, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3krlA (A:)
gvdykykqkpkyqvrwkiiesyegnsytfidptqlpynekwefprnnlqfgktlgagafg
kvveatafglgkedavlkvavkmlkstahadekealmselkimshlgqhenivnllgact
hggpvlviteyccygdllnflrrkrppgleysynpshnpeeqlssrdllhfssqvaqgma
flaskncihrdvaarnvlltnghvakigdfglardimndsnyivkgnarlpvkwmapesi
fdcvytvqsdvwsygillweifslglnpypgilvnskfyklvkdgyqmaqpafapkniys
imqacwalepthrptfqqicsflqeqaqedrrerd
Sequence, based on observed residues (ATOM records): (download)
>3krlA (A:)
kyqvrwkiipynekwefprnnlqfgktlgagafgkvveatafglgkedavlkvavkmlks
taadekealmselkimshlgqhenivnllgacthggpvlviteyccygdllnflrrkrql
ssrdllhfssqvaqgmaflaskncihrdvaarnvlltnghvakigdfglardimndsnyi
vkgarlpvkwmapesifdcvytvqsdvwsygillweifslglnpypgilvnskfyklvkd
gyqmaqpafapkniysimqacwalepthrptfqqicsflqe