PDB entry 3js2
View 3js2 on RCSB PDB site
Description: Crystal structure of minimal kinase domain of fibroblast growth factor receptor 1 in complex with 5-(2-thienyl)nicotinic acid
Class: transferase
Keywords: fibroblast growth factor, receptor tyrosine kinase, inhibitor, thienyl nicotinic acid, Alternative splicing, ATP-binding, Chromosomal rearrangement, Craniosynostosis, Disease mutation, Disulfide bond, Dwarfism, Glycoprotein, Heparin-binding, Hypogonadotropic hypogonadism, Immunoglobulin domain, Kallmann syndrome, Kinase, Membrane, Nucleotide-binding, Phosphoprotein, Polymorphism, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on
2009-09-09, released
2010-02-23
The last revision prior to the SCOPe 2.05 freeze date was dated
2010-03-02, with a file datestamp of
2010-02-26.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.216
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Basic fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, FGFBR, FLG, FLT2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3js2a_ - Chain 'B':
Compound: Basic fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, FGFBR, FLG, FLT2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3js2b_ - Heterogens: VM1, PO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3js2A (A:)
mghhhhhhmagvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrv
tkvavkmlksdatekdlsdlisememmkmigkhkniinllgactqdgplyviveyaskgn
lreylqarrppgleysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarn
vlvtednvmkiadfglardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgv
llweiftlggspypgvpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfk
qlvedldrivaltsnqe
Sequence, based on observed residues (ATOM records): (download)
>3js2A (A:)
elpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkmlksdatek
dlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrppglhn
peeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfglardihh
idyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypgvpveelf
kllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivaltsnqe
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3js2B (B:)
mghhhhhhmagvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrv
tkvavkmlksdatekdlsdlisememmkmigkhkniinllgactqdgplyviveyaskgn
lreylqarrppgleysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarn
vlvtednvmkiadfglardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgv
llweiftlggspypgvpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfk
qlvedldrivaltsnqe
Sequence, based on observed residues (ATOM records): (download)
>3js2B (B:)
gvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkmlks
datekdlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrp
peqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfglardihhi
dyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypgvpveelfk
llkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivalts