PDB entry 3inh
View 3inh on RCSB PDB site
Description: Bace1 with the aminohydantoin Compound R-58
Class: hydrolase
Keywords: Bace1, xray, inhibitor, Alternative splicing, Aspartyl protease, Disulfide bond, Glycoprotein, Hydrolase, Membrane, Polymorphism, Protease, Transmembrane, Zymogen
Deposited on
2009-08-12, released
2010-03-02
The last revision prior to the SCOPe 2.05 freeze date was dated
2010-03-02, with a file datestamp of
2010-02-26.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.211
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Beta-secretase 1
Species: Homo sapiens [TaxId:9606]
Gene: BACE1, BACE, KIAA1149
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3inha_ - Heterogens: 569, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3inhA (A:)
etdeepeepgrrgsfvemvdnlrgksgqgyyvemtvgsppqtlnilvdtgssnfavgaap
hpflhryyqrqlsstyrdlrkgvyvpytqgkwegelgtdlvsiphgpnvtvraniaaite
sdkffingsnwegilglayaeiarpddslepffdslvkqthvpnlfslqlcgagfplnqs
evlasvggsmiiggidhslytgslwytpirrewyyeviivrveingqdlkmdckeynydk
sivdsgttnlrlpkkvfeaavksikaasstekfpdgfwlgeqlvcwqagttpwnifpvis
lylmgevtnqsfritilpqqylrpvedvatsqddcykfaisqsstgtvmgavimegfyvv
fdrarkrigfavsachvhdefrtaavegpfvtldmedcgynipqtdesthhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3inhA (A:)
sfvemvdnlrgksgqgyyvemtvgsppqtlnilvdtgssnfavgaaphpflhryyqrqls
styrdlrkgvyvpykwegelgtdlvsiphgpnvtvraniaaitesdkffingsnwegilg
layaeiarpddslepffdslvkqthvpnlfslqlcgagflasvggsmiiggidhslytgs
lwytpirrewyyeviivrveingqdlkmdckeynydksivdsgttnlrlpkkvfeaavks
ikaasstekfpdgfwlgeqlvcwqagttpwnifpvislylmgevtnqsfritilpqqylr
pcykfaisqsstgtvmgavimegfyvvfdrarkrigfavsachvhdefrtaavegpfvtl
dcgyni