PDB entry 3hxd
View 3hxd on RCSB PDB site
Description: Engineered RabGGTase in complex with a peptidomimetic inhibitor (compound 9)
Class: transferase
Keywords: protein prenylation inhibition, TRANSFERASE
Deposited on
2009-06-20, released
2009-09-08
The last revision prior to the SCOPe 2.04 freeze date was dated
2009-12-29, with a file datestamp of
2009-12-24.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: 0.174
AEROSPACI score: 0.5
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Geranylgeranyl transferase type-2 subunit alpha
Species: Rattus norvegicus [TaxId:10116]
Database cross-references and differences (RAF-indexed):
- Chain 'B':
Compound: Geranylgeranyl transferase type-2 subunit beta
Species: Rattus norvegicus [TaxId:10116]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d3hxdb_ - Heterogens: ZN, CA, BD7, HOH
PDB Chain Sequences:
- Chain 'A':
No sequence available.
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3hxdB (B:)
mgtqqkdvtiksdapdtlllekhadyiasygskkddyeycmseylrmsgvywgltvmdlm
gqlhrmnkeeilvfikscqhecggvsasighdphllytlsavqiltlydsihvinvdkvv
ayvqslqkedgsfagdiwgeidtrfsfcavatlallgkldainvekaiefvlscmnfdgg
fgcrpgseshagqiycctgflaitsqlhqvnsdllgwwlcerqlpsgglngrpeklpdvc
yswwvlaslkiigrlhwidreklrsfilacqdeetggfadrpgdmvdpfhtlfgiaglsl
lgeeqikpvspvfcmpeevlqrvnvqpelvs
Sequence, based on observed residues (ATOM records): (download)
>3hxdB (B:)
qkdvtiksdapdtlllekhadyiasygsdyeycmseylrmsgvywgltvmdlmgqlhrmn
keeilvfikscqhecggvsasighdphllytlsavqiltlydsihvinvdkvvayvqslq
kedgsfagdiwgeidtrfsfcavatlallgkldainvekaiefvlscmnfdggfgcrpgs
eshagqiycctgflaitsqlhqvnsdllgwwlcerqlpsgglngrpeklpdvcyswwvla
slkiigrlhwidreklrsfilacqdeetggfadrpgdmvdpfhtlfgiaglsllgeeqik
pvspvfcmpeevlqrvnvqpelvs