PDB entry 3h9o

View 3h9o on RCSB PDB site
Description: Phosphoinositide-dependent protein kinase 1 (PDK-1) in complex with compound 9
Class: transferase
Keywords: PDK-1, kinase, protein structure, X-ray crysatllography, Alternative splicing, ATP-binding, Cytoplasm, Membrane, Nucleotide-binding, Phosphoprotein, Serine/threonine-protein kinase, Transferase
Deposited on 2009-04-30, released 2009-08-25
The last revision prior to the SCOPe 2.03 freeze date was dated 2009-08-25, with a file datestamp of 2009-08-21.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: 0.211
AEROSPACI score: 0.35 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: 3-phosphoinositide-dependent protein kinase 1
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.03: d3h9oa_
  • Heterogens: 9BD, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3h9oA (A:)
    gpmdgtaaeprpgagslqhaqpppqprkkrpedfkfgkilgegsfstvvlarelatsrey
    aikilekrhiikenkvpyvtrerdvmsrldhpffvklyftfqddeklyfglsyakngell
    kyirkigsfdetctrfytaeivsaleylhgkgiihrdlkpenillnedmhiqitdfgtak
    vlspeskqaransfvgtaqyvspellteksackssdlwalgciiyqlvaglppfragney
    lifqkiikleydfpekffpkardlvekllvldatkrlgceemegygplkahpffesvtwe
    nlhqqtppklt
    

    Sequence, based on observed residues (ATOM records): (download)
    >3h9oA (A:)
    rkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerdvm
    srldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsale
    ylhgkgiihrdlkpenillnedmhiqitdfgtakvlssfvgtaqyvspellteksackss
    dlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlvekllvldatk
    rlgceemegygplkahpffesvtwenlhqqtppklt