PDB entry 3gi3
View 3gi3 on RCSB PDB site
Description: Crystal structure of a N-Phenyl-N'-Naphthylurea analog in complex with p38 MAP kinase
Class: transferase
Keywords: two lobe kinase structure, N-lobe beta-sheet, C-lobe alpha-helix, Alternative splicing, ATP-binding, Cytoplasm, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Polymorphism, Serine/threonine-protein kinase, Transferase
Deposited on
2009-03-05, released
2009-10-20
The last revision prior to the SCOPe 2.05 freeze date was dated
2009-10-20, with a file datestamp of
2009-10-16.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.23
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2
Database cross-references and differences (RAF-indexed):
- Uniprot Q16539
- conflict (47)
- conflict (169)
Domains in SCOPe 2.05: d3gi3a_ - Heterogens: B10, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3gi3A (A:)
msqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktghrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfylarhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3gi3A (A:)
rptfyrqelnktiwevperyqnlspvsvcaafdtktghrvavkklsrpfqsiihakrtyr
elrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltddhvqfl
iyqilrglkyihsadiihrdlkpsnlavnedcelkildfyvatrwyrapeimlnwmhynq
tvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqsl
tqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadp
ydqsfesrdllidewksltydevisfvppp