PDB entry 3ggu
View 3ggu on RCSB PDB site
Description: HIV PR drug resistant patient's variant in complex with darunavir
Class: hydrolase
Keywords: darunvir, resistance, mutation score, HIV protease, TMC-114, HYDROLASE
Deposited on
2009-03-02, released
2009-08-11
The last revision prior to the SCOPe 2.04 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-25.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.206
AEROSPACI score: 0.48
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Protease
Species: Human immunodeficiency virus type 1 (BRU ISOLATE) [TaxId:11686]
Gene: Gag-Pol, pol
Database cross-references and differences (RAF-indexed):
- Uniprot P03367 (0-98)
- engineered (9)
- engineered (12)
- engineered (15)
- engineered (32)
- engineered (35-36)
- engineered (38)
- engineered (44-45)
- engineered (53-54)
- engineered (61-62)
- engineered (70)
- engineered (72)
- engineered (81)
- engineered (83)
- engineered (88-89)
- engineered (92)
Domains in SCOPe 2.04: d3ggua_ - Chain 'B':
Compound: Protease
Species: Human immunodeficiency virus type 1 (BRU ISOLATE) [TaxId:11686]
Gene: Gag-Pol, pol
Database cross-references and differences (RAF-indexed):
- Uniprot P03367 (0-98)
- engineered (9)
- engineered (12)
- engineered (15)
- engineered (32)
- engineered (35-36)
- engineered (38)
- engineered (44-45)
- engineered (53-54)
- engineered (61-62)
- engineered (70)
- engineered (72)
- engineered (81)
- engineered (83)
- engineered (88-89)
- engineered (92)
Domains in SCOPe 2.04: d3ggub_ - Heterogens: 017, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>3gguA (A:)
pqitlwqrpivtvkiegqlkealldtgaddtvfeeltlsgrwkprliggiggfvrvrqyd
qvpieicghkvidtvlvgptptnvigrnvmtqlgctlnf
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>3gguB (B:)
pqitlwqrpivtvkiegqlkealldtgaddtvfeeltlsgrwkprliggiggfvrvrqyd
qvpieicghkvidtvlvgptptnvigrnvmtqlgctlnf