PDB entry 3g0w

View 3g0w on RCSB PDB site
Description: Crystal structure of the rat androgen receptor ligand binding domain complex with an n-aryl-oxazolidin 2-imine inhibitor
Class: hormone
Keywords: ANDROGEN RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN, Disease mutation, DNA-binding, Lipid-binding, Metal-binding, Nucleus, Phosphoprotein, Receptor, Steroid-binding, Transcription, Ubl conjugation, Zinc, Zinc-finger, HORMONE/GROWTH FACTOR COMPLEX
Deposited on 2009-01-29, released 2009-04-28
The last revision prior to the SCOPe 2.08 freeze date was dated 2009-05-26, with a file datestamp of 2009-05-22.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: 0.201
AEROSPACI score: 0.45 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Androgen receptor
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Ar, Nr3c4
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d3g0wa_
  • Heterogens: LGB, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3g0wA (A:)
    gshmiegyecqpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwa
    kalpgfrnlhvddqmaviqyswmglmvfamgwrsftnvnsrmlyfapdlvfneyrmhksr
    mysqcvrmrhlsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeld
    riiackrknptscsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeii
    svqvpkilsgkvkpiyfhtq
    

    Sequence, based on observed residues (ATOM records): (download)
    >3g0wA (A:)
    qpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnlh
    vddqmaviqyswmglmvfamgwrsftnvnsrmlyfapdlvfneyrmhksrmysqcvrmrh
    lsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiackrknp
    tscsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkilsg
    kvkpiyfht