PDB entry 3g0w
View 3g0w on RCSB PDB site
Description: Crystal structure of the rat androgen receptor ligand binding domain complex with an n-aryl-oxazolidin 2-imine inhibitor
Class: hormone
Keywords: ANDROGEN RECEPTOR, STEROID RECEPTOR, NUCLEAR RECEPTOR, TRANSCRIPTION REGULATION, LIGAND-BINDING DOMAIN, Disease mutation, DNA-binding, Lipid-binding, Metal-binding, Nucleus, Phosphoprotein, Receptor, Steroid-binding, Transcription, Ubl conjugation, Zinc, Zinc-finger, HORMONE/GROWTH FACTOR COMPLEX
Deposited on
2009-01-29, released
2009-04-28
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-05-26, with a file datestamp of
2009-05-22.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: 0.201
AEROSPACI score: 0.45
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Androgen receptor
Species: Rattus norvegicus [TaxId:10116]
Gene: Ar, Nr3c4
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3g0wa_ - Heterogens: LGB, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3g0wA (A:)
gshmiegyecqpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwa
kalpgfrnlhvddqmaviqyswmglmvfamgwrsftnvnsrmlyfapdlvfneyrmhksr
mysqcvrmrhlsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeld
riiackrknptscsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeii
svqvpkilsgkvkpiyfhtq
Sequence, based on observed residues (ATOM records): (download)
>3g0wA (A:)
qpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnlh
vddqmaviqyswmglmvfamgwrsftnvnsrmlyfapdlvfneyrmhksrmysqcvrmrh
lsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiackrknp
tscsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkilsg
kvkpiyfht