PDB entry 3fzk
View 3fzk on RCSB PDB site
Description: Crystal Structures of Hsc70/Bag1 in Complex with Small Molecule Inhibitors
Class: chaperone
Keywords: HSP70, HSC70, BAG1, heat shock, chaperone, protein folding, adenosine, nucleotide, nucleotide exchange factor, small molecule inhibitor, ATP-binding, nucleotide-binding, stress response, apoptosis
Deposited on
2009-01-26, released
2009-03-17
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-03-31, with a file datestamp of
2009-03-27.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.222
AEROSPACI score: 0.37
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Heat shock cognate 71 kDa protein
Species: Homo sapiens [TaxId:9606]
Gene: HSPA8, HSC70, HSP73, HSPA10
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3fzka1, d3fzka2 - Chain 'B':
Compound: BAG family molecular chaperone regulator 1
Species: Homo sapiens [TaxId:9606]
Gene: BAG1, HAP
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3fzkb1, d3fzkb2 - Heterogens: TRS, CL, 3BK, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3fzkA (A:)
yfqgpavgidlgttyscvgvfqhgkveiiandqgnrttpsyvaftdterligdaaknqva
mnptntvfdakrligrrfddavvqsdmkhwpfmvvndagrpkvqveykgetksfypeevs
smvltkmkeiaeaylgktvtnavvtvpayfndsqrqatkdagtiaglnvlriineptaaa
iaygldkkvgaernvlifdlgggtfdvsiltiedgifevkstagdthlggedfdnrmvnh
fiaefkrkhkkdisenkravrrlrtacerakrtlssstqasieidslyegidfytsitra
rfeelnadlfrgtldpvekalrdakldksqihdivlvggstripkiqkllqdffngkeln
ksinpdeavaygaavqaails
Sequence, based on observed residues (ATOM records): (download)
>3fzkA (A:)
pavgidlgttyscvgvfqhgkveiiandqgnrttpsyvaftdterligdaaknqvamnpt
ntvfdakrligrrfddavvqsdmkhwpfmvvndagrpkvqveykgetksfypeevssmvl
tkmkeiaeaylgktvtnavvtvpayfndsqrqatkdagtiaglnvlriineptaaaiayg
ldkkvgaernvlifdlgggtfdvsiltiedgifevkstagdthlggedfdnrmvnhfiae
fkrkhkkdisenkravrrlrtacerakrtlssstqasieidslyegidfytsitrarfee
lnadlfrgtldpvekalrdakldksqihdivlvggstripkiqkllqdffngkelnksin
pdeavaygaavqaails
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3fzkB (B:)
gnspqeevelkklkhleksvekiadqleelnkeltgiqqgflpkdlqaealckldrrvka
tieqfmkileeidtlilpenfkdsrlkrkglvkkvqaflaecdtveqnicqete
Sequence, based on observed residues (ATOM records): (download)
>3fzkB (B:)
gnspqeevelkklkhleksvekiadqleelnkeltgiqqgflpkdlqaealckldrrvka
tieqfmkileeidtlilpenfkdsrlkrkglvkkvqaflaecdtveqnicq