PDB entry 3fv8
View 3fv8 on RCSB PDB site
Description: JNK3 bound to piperazine amide inhibitor, SR2774.
Class: transferase
Keywords: JNK3, protein-inhibitor complex, Alternative splicing, ATP-binding, Chromosomal rearrangement, Cytoplasm, Epilepsy, Kinase, Nucleotide-binding, Phosphoprotein, Serine/threonine-protein kinase, Transferase
Deposited on
2009-01-15, released
2009-04-07
The last revision prior to the SCOPe 2.06 freeze date was dated
2009-06-30, with a file datestamp of
2009-06-26.
Experiment type: XRAY
Resolution: 2.28 Å
R-factor: 0.204
AEROSPACI score: 0.35
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 10
Species: Homo sapiens [TaxId:9606]
Gene: JNK3, JNK3A, MAPK10, PRKM10
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3fv8a_ - Heterogens: JK3, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3fv8A (A:)
mskskvdnqfysvevgdstftvlkryqnlkpigsgaqgivcaaydavldrnvaikklsrp
fqnqthakrayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviq
meldhermsyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartagtsf
mmtpyvvtryyrapevilgmgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieq
lgtpcpefmkklqptvrnyvenrpkyagltfpklfpdslfpadsehnklkasqardllsk
mlvidpakrisvddalqhpyinvwydpaxxxxxderehtieewkeliykevmnse
Sequence, based on observed residues (ATOM records): (download)
>3fv8A (A:)
nqfysvevgdstftvlkryqnlkpigsgaqgivcaaydavldrnvaikklsrpfqnqtha
krayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviqmeldher
msyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglarvtryyrapevilg
mgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieqlgtpcpefmkklqptvrny
venrpkyagltfpklfpdslfpadsehnklkasqardllskmlvidpakrisvddalqhp
yinvwydpaxxxxxderehtieewkeliykevmn