PDB entry 3fi4
View 3fi4 on RCSB PDB site
Description: P38 kinase crystal structure in complex with RO4499
Class: signaling protein, transferase
Keywords: P38; MAP KINASE; SERINE/THREONINE KINASE, Alternative splicing, ATP-binding, Cytoplasm, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Polymorphism, Serine/threonine-protein kinase, Transferase, SIGNALING PROTEIN
Deposited on
2008-12-10, released
2009-12-22
The last revision prior to the SCOPe 2.07 freeze date was dated
2009-12-22, with a file datestamp of
2009-12-18.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.212
AEROSPACI score: 0.39
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: CSBP, CSBP1, CSBP2, CSPB1, MAPK14, MXI2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d3fi4a_ - Heterogens: FI4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3fi4A (A:)
mrgshhhhhhgsmsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktgl
rvavkklskpfqsiihakrtyrelrllkhmkhenviglldvftparsleefndvylvthl
mgadlnnivkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkild
fglarhtddemtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdh
idqlklilrlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekm
lvldsdkritaaqalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisf
vpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3fi4A (A:)
erptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklskpfqsii
hakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnniddhvqfl
iyqilrglkyihsadiihrdlkpsnlavnedcelkildfgltddemtgyvatrwyrapei
mlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkisse
sarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhd
pddepvadpydqsfesrdllidewksltydevisfvppp