PDB entry 3fhr
View 3fhr on RCSB PDB site
Description: High resolution crystal structure of mitogen-activated protein kinase-activated protein kinase 3 (MK3)-inhibitor complex
Class: transferase
Keywords: Kinase-inhibitor complex, ATP-binding, Cytoplasm, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Polymorphism, Serine/threonine-protein kinase, Transferase
Deposited on
2008-12-10, released
2009-12-15
The last revision prior to the SCOPe 2.03 freeze date was dated
2009-12-15, with a file datestamp of
2009-12-11.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.228
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: MAP kinase-activated protein kinase 3
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3fhra_ - Heterogens: P4O, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3fhrA (A:)
mahhhhhhssglevlfqgpepkkyavtddyqlskqvlglgvngkvlecfhrrtgqkcalk
llydspkarqevdhhwqasggphivcildvyenmhhgkrclliimecmeggelfsriqer
gdqaftereaaeimrdigtaiqflhshniahrdvkpenllytskekdavlkltdfgfake
ttqnalqtpcytpyyvapevlgpekydkscdmwslgvimyillcgfppfysntgqaispg
mkrrirlgqygfpnpewsevsedakqlirlllktdpterltitqfmnhpwinqsmvvpqt
plhtarvlqedkdhwdevkeemtsalatmrvdydqv
Sequence, based on observed residues (ATOM records): (download)
>3fhrA (A:)
epkkyavtddyqlskqvlglgvngkvlecfhrrtgqkcalkllydspkarqevdhhwqas
ggphivcildvyenmhhgkrclliimecmeggelfsriqerdqaftereaaeimrdigta
iqflhshniahrdvkpenllytskekdavlkltdfgfaketekydkscdmwslgvimyil
lcgfppfgfpnpewsevsedakqlirlllktdpterltitqfmnhpwinqsmvvpqtplh
tarvlqedkdhwdevkeemtsalatmrvdydqv