PDB entry 3f82
View 3f82 on RCSB PDB site
Description: Crystal structure of the tyrosine kinase domain of the hepatocyte growth factor receptor C-MET in complex with N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
Class: transferase
Keywords: Alternative splicing, RECEPTOR TYROSINE KINASE, SIGNAL TRANSDUCTION, GRB2, SHC, ATP-BINDING, GLYCOPROTEIN, MEMBRANE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PROTO-ONCOGENE, TRANSFERASE, TRANSMEMBRANE, TYROSINE-PROTEIN KINASE
Deposited on
2008-11-11, released
2009-03-31
The last revision prior to the SCOPe 2.05 freeze date was dated
2009-03-31, with a file datestamp of
2009-03-27.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.183
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3f82a_ - Heterogens: 353, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3f82A (A:)
gantvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkih
cavkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlr
nfirnethnptvkdligfglqvakgmkflaskkfvhrdlaarncmldekftvkvadfgla
rdmydkefdsvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypd
vntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfig
ehyvhvnatyvnvk
Sequence, based on observed residues (ATOM records): (download)
>3f82A (A:)
lsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtllkihcavkslnrgevsq
fltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrnfirnethnptvkdlig
fglqvakgmkflaskkfvhrdlaarncmldekftvkvadfgklpvkwmaleslqtqkftt
ksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpeycpdplyevmlkcwhp
kaemrpsfselvsrisaifstfigehyvhvnatyvnvk