PDB entry 3eyg

View 3eyg on RCSB PDB site
Description: Crystal structures of JAK1 and JAK2 inhibitor complexes
Class: transferase
Keywords: JAK kinase, ATP-binding, Kinase, Nucleotide-binding, Phosphoprotein, SH2 domain, Transferase, Tyrosine-protein kinase
Deposited on 2008-10-20, released 2009-02-03
The last revision prior to the SCOPe 2.08 freeze date was dated 2009-12-29, with a file datestamp of 2009-12-24.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.171
AEROSPACI score: 0.48 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Tyrosine-protein kinase
    Species: Homo sapiens [TaxId:9606]
    Gene: JAK1, hCG_22179
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d3eyga_
  • Heterogens: MI1, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3eygA (A:)
    vdpthfekrflkrirdlgeghfgkvelcrydpegdntgeqvavkslkpesggnhiadlkk
    eieilrnlyhenivkykgictedggngiklimeflpsgslkeylpknknkinlkqqlkya
    vqickgmdylgsrqyvhrdlaarnvlvesehqvkigdfgltkaietdkeyytvkddrdsp
    vfwyapeclmqskfyiasdvwsfgvtlhelltycdsdsspmalflkmigpthgqmtvtrl
    vntlkegkrlpcppncpdevyqlmrkcwefqpsnrtsfqnliegfeallk
    

    Sequence, based on observed residues (ATOM records): (download)
    >3eygA (A:)
    vdpthfekrflkrirdlgeghfgkvelcrydpegdntgeqvavkslkphiadlkkeieil
    rnlyhenivkykgictengiklimeflpsgslkeylpknknkinlkqqlkyavqickgmd
    ylgsrqyvhrdlaarnvlvesehqvkigdfgltkaietdkeyytvkddrdspvfwyapec
    lmqskfyiasdvwsfgvtlhelltycdsdsspmalflkmigpthgqmtvtrlvntlkegk
    rlpcppncpdevyqlmrkcwefqpsnrtsfqnliegfeallk