PDB entry 3eta
View 3eta on RCSB PDB site
Description: Kinase domain of insulin receptor complexed with a pyrrolo pyridine inhibitor
Class: signaling protein, transferase
Keywords: ATP-binding, Carbohydrate metabolism, Cleavage on pair of basic residues, Diabetes mellitus, Disease mutation, Glycoprotein, Kinase, Membrane, Nucleotide-binding, Phosphoprotein, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase, SIGNALING PROTEIN
Deposited on
2008-10-07, released
2009-05-26
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 2.6 Å
R-factor: 0.203
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: insulin receptor, kinase domain
Species: Homo sapiens [TaxId:9606]
Gene: INSR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3etaa_ - Chain 'B':
Compound: insulin receptor, kinase domain
Species: Homo sapiens [TaxId:9606]
Gene: INSR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3etab_ - Heterogens: 351, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3etaA (A:)
mkkghhhhhhgevsrekitllrelgqgsfgmvyegnardiikgeaetrvavktvnesasl
rerieflneasvmkgftchhvvrllgvvskgqptlvvmelmahgdlksylrslrpeaenn
pgrppptlqemiqmaaeiadgmaylnakkfvhrdlaarncmvahdftvkigdfgmtrdiy
etdyyrkggkgllpvrwmapeslkdgvfttssdmwsfgvvlweitslaeqpyqglsneqv
lkfvmdggyldqpdncpervtdlmrmcwqfnpkmrptfleivnllkddlhpsfpevsffh
seenkapeseelemefe
Sequence, based on observed residues (ATOM records): (download)
>3etaA (A:)
evsrekitllrelgqgsfgmvyegnardiikgeaetrvavktvnesaslrerieflneas
vmkgftchhvvrllgvvskgqptlvvmelmahgdlksylrslrpeaennpgrppptlqem
iqmaaeiadgmaylnakkfvhrdlaarncmvahdftvkigdfgmtrdiyetdyyrkgkgl
lpvrwmapeslkdgvfttssdmwsfgvvlweitslaeqpyqglsneqvlkfvmdggyldq
pdncpervtdlmrmcwqfnpkmrptfleivnllkddlhpsfpevsffhseenk
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3etaB (B:)
mkkghhhhhhgevsrekitllrelgqgsfgmvyegnardiikgeaetrvavktvnesasl
rerieflneasvmkgftchhvvrllgvvskgqptlvvmelmahgdlksylrslrpeaenn
pgrppptlqemiqmaaeiadgmaylnakkfvhrdlaarncmvahdftvkigdfgmtrdiy
etdyyrkggkgllpvrwmapeslkdgvfttssdmwsfgvvlweitslaeqpyqglsneqv
lkfvmdggyldqpdncpervtdlmrmcwqfnpkmrptfleivnllkddlhpsfpevsffh
seenkapeseelemefe
Sequence, based on observed residues (ATOM records): (download)
>3etaB (B:)
evsrekitllrelgqgsfgmvyegnardiikgeaetrvavktvnesaslrerieflneas
vmkgftchhvvrllgvvskgqptlvvmelmahgdlksylrslrpeaennpgrppptlqem
iqmaaeiadgmaylnakkfvhrdlaarncmvahdftvkigdfgmtrdiyetdyyrkkgll
pvrwmapeslkdgvfttssdmwsfgvvlweitslaeqpyqglsneqvlkfvmdggyldqp
dncpervtdlmrmcwqfnpkmrptfleivnllkddlhpsfpevsffhseenk