PDB entry 3et3
View 3et3 on RCSB PDB site
Description: Structure of PPARgamma with 3-[5-Methoxy-1-(4-methoxy-benzenesulfonyl)-1H-indol-3-yl]-propionic acid
Class: transcription
Keywords: PPAR, PPARg, PPARgamma, Drug Discovery, Diabetes, adiponectin, metabolic disease, fragment-based drug discovery, scaffold-based drug discovery, Activator, Alternative splicing, Diabetes mellitus, Disease mutation, DNA-binding, Metal-binding, Nucleus, Obesity, Phosphoprotein, Polymorphism, Receptor, Transcription, Transcription regulation, Zinc, Zinc-finger, Acyltransferase, Chromosomal rearrangement, Proto-oncogene, Transferase, Ubl conjugation
Deposited on
2008-10-06, released
2009-02-17
The last revision prior to the SCOPe 2.05 freeze date was dated
2009-02-17, with a file datestamp of
2009-02-13.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: 0.182
AEROSPACI score: 0.48
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Peroxisome proliferator-activated receptor gamma
Species: Homo sapiens [TaxId:9606]
Gene: PPARG, NR1C3
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3et3a_ - Chain 'P':
Compound: steroid receptor coactivator 1
Species: Homo sapiens [TaxId:9606]
Gene: NCOA1, SRC1
Database cross-references and differences (RAF-indexed):
- Heterogens: ET1, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3et3A (A:)
mgsshhhhhhssglvprgshmesadlralakhlydsyiksfpltkakarailtgkttdks
pfviydmnslmmgedkikfkhitplqeqskevairifqgcqfrsveavqeiteyaksipg
fvnldlndqvtllkygvheiiytmlaslmnkdgvlisegqgfmtreflkslrkpfgdfme
pkfefavkfnalelddsdlaifiaviilsgdrpgllnvkpiediqdnllqalelqlklnh
pessqlfakllqkmtdlrqivtehvqllqvikktetdmslhpllqeiykdly
Sequence, based on observed residues (ATOM records): (download)
>3et3A (A:)
mesadlralakhlydsyiksfpltkakarailtgkttdkspfviydmnslmmgedkikev
airifqgcqfrsveavqeiteyaksipgfvnldlndqvtllkygvheiiytmlaslmnkd
gvlisegqgfmtreflkslrkpfgdfmepkfefavkfnalelddsdlaifiaviilsgdr
pgllnvkpiediqdnllqalelqlklnhpessqlfakllqkmtdlrqivtehvqllqvik
ktetdmslhpllqeiykdly
- Chain 'P':
No sequence available.