PDB entry 3ekk
View 3ekk on RCSB PDB site
Description: Insulin receptor kinase complexed with an inhibitor
Class: transferase
Keywords: insulin, tyrosine kinase, ATP-binding, Carbohydrate metabolism, Cleavage on pair of basic residues, Diabetes mellitus, Disease mutation, Glycoprotein, Kinase, Membrane, Nucleotide-binding, Phosphoprotein, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on
2008-09-19, released
2008-12-23
The last revision prior to the SCOPe 2.02 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.207
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Insulin receptor
Species: Homo sapiens [TaxId:9606]
Gene: INSR
Database cross-references and differences (RAF-indexed):
- Uniprot P06213
- engineered (4)
- engineered (155)
- see remark 999 (274)
Domains in SCOPe 2.02: d3ekka_ - Heterogens: GS2, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3ekkA (A:)
gvfpssvyvpdewevsrekitllrelgqgsfgmvyegnardiikgeaetrvavktvnesa
slrerieflneasvmkgftchhvvrllgvvskgqptlvvmelmahgdlksylrslrpeae
nnpgrppptlqemiqmaaeiadgmaylnakkfvhrnlaarncmvahdftvkigdfgmtrd
iyetdyyrkggkgllpvrwmapeslkdgvfttssdmwsfgvvlweitslaeqpyqglsne
qvlkfvmdggyldqpdncpervtdlmrmcwqfnpnmrptfleivnllkddlhpsfpevsf
fhseenk
Sequence, based on observed residues (ATOM records): (download)
>3ekkA (A:)
pssvyvpdewevsrekitllrelgqgsfgmvyegnardiikgeaetrvavktvnesaslr
erieflneasvmkgftchhvvrllgvvskgqptlvvmelmahgdlksylrslrpeaennp
grppptlqemiqmaaeiadgmaylnakkfvhrnlaarncmvahdftvkigdfllpvrwma
peslkdgvfttssdmwsfgvvlweitslaeqpyqglsneqvlkfvmdggyldqpdncper
vtdlmrmcwqfnpnmrptfleivnllkddlhpsfpevsffhseen