PDB entry 3e92
View 3e92 on RCSB PDB site
Description: Crystal Structure of P38 Kinase in Complex with A Biaryl Amide Inhibitor
Class: transferase
Keywords: P38, SERINE/THREONINE PROTEIN KINASE, MAP KINASE, ATP-binding, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Serine/threonine-protein kinase, TRANSFERASE
Deposited on
2008-08-21, released
2008-09-30
The last revision prior to the SCOPe 2.01 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.174
AEROSPACI score: 0.47
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d3e92a_ - Heterogens: G6A, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3e92A (A:)
mkkghhlhhhgmsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglr
vavkklsrpfqsiihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlm
gadlnnivkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildf
glarhtddemtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhi
dqlklilrlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekml
vldsdkritaaqalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfv
pppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3e92A (A:)
qerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsi
ihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkl
tddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglahtddemtgyv
atrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpg
aellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqal
ahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvppp