PDB entry 3dt1
View 3dt1 on RCSB PDB site
Description: P38 Complexed with a quinazoline inhibitor
Class: transferase
Keywords: Kinase Inhibitor complex, Alternative splicing, ATP-binding, Cytoplasm, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Polymorphism, Serine/threonine-protein kinase, Transferase
Deposited on
2008-07-14, released
2008-10-14
The last revision prior to the SCOPe 2.03 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 2.8 Å
R-factor: 0.214
AEROSPACI score: 0.25
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3dt1a_ - Heterogens: P40, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3dt1A (A:)
mgsshhhhhhssglvprgshmlemsqerptfyrqelnktiwevperyqnlspvgsgaygs
vcaafdtktglrvavkklsrpfqsiihakrtyrelrllkhmkhenviglldvftparsle
efndvylvthlmgadlnnivkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnla
vnedcelkildfglarhtddemtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaell
tgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiga
nplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadpydqsfesrdllidew
ksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3dt1A (A:)
hmlemsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkkls
rpfqsiihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnni
vkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtd
demtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklil
rlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkr
itaaqalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvppp